SCHEMBL6169112

SCHEMBL6169112

N#Cc1cccc(C#N)c1Oc1cn[nH]c1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
MAPT P10636 2/20 0.38
NPSR1 Q6W5P4 1/20 0.38
HTT P42858 1/20 0.34
PRKCQ Q04759 1/20 0.34
PDE4B Q07343 3/20 0.33
AR P10275 2/20 0.33
DYRK1A Q13627 1/20 0.33
POLB P06746 1/20 0.33
GAA P10253 1/20 0.33
CYP19A1 P11511 1/20 0.33
PIN1 Q13526 1/20 0.33
MAP2K1 Q02750 1/20 0.33
AKT1 P31749 1/20 0.32
AKT2 P31751 1/20 0.32
KDM4C Q9H3R0 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6216924 0.81 POLB (0.54) ALDH1A1SMN1; SMN2PDE4BARPOLB
SCHEMBL24210848 0.73 KCNH2 (0.40) SMN1; SMN2NPSR1PDE4BARAKT1
SCHEMBL4733455 0.71 CYP19A1 (0.53) ALDH1A1SMN1; SMN2MAPTPDE4BPOLB
SCHEMBL11332971 0.71 MAPT (0.48) SMN1; SMN2MAPTNPSR1PDE4BAR
SCHEMBL2750417 0.71 MAPT (0.44) ALDH1A1SMN1; SMN2MAPTNPSR1AR
SCHEMBL16969031 0.69 AR (0.51) ALDH1A1SMN1; SMN2MAPTNPSR1HTT
SCHEMBL509280 0.68 KCNH2 (0.41) CYP19A1KDM4C
SCHEMBL28439643 0.68 MAPT (0.43) ALDH1A1SMN1; SMN2MAPTNPSR1POLB
SCHEMBL3251181 0.67 CYP1A2 (0.43) ALDH1A1SMN1; SMN2MAPTNPSR1HTT
SCHEMBL2753440 0.67 MAPT (0.42) ALDH1A1SMN1; SMN2MAPTNPSR1AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546132-A1 PYRAZOLE DERIVATIVES AS REVERSE TRANSCRIPTASE INHIBITORS Pfizer Limited (GB) 2005-06-29 EP disclosed
WO-2004029042-A1 PYRAZOLE DERIVATIVES AS REVERSE TRANSCRIPTASE INHIBITORS PFIZER LIMITED (GB) 2004-04-08 WO disclosed