SCHEMBL6169664

SCHEMBL6169664

c1ccc(C(c2ccccc2)N2CCC3(CCc4ccccc43)CC2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 10/20 0.56
CYP2C9 P11712 2/20 0.56
CYP2C19 P33261 2/20 0.56
CYP2D6 P10635 2/20 0.56
ALDH1A1 P00352 1/20 0.56
TP53 P04637 1/20 0.56
CYP1A2 P05177 1/20 0.56
CYP3A4 P08684 1/20 0.56
TSHR P16473 1/20 0.56
OPRM1 P35372 8/20 0.51
OPRK1 P41145 7/20 0.51
OPRL1 P41146 7/20 0.51
OPRD1 P41143 6/20 0.51
SLC18A3 Q16572 3/20 0.50
USP2 O75604 1/20 0.49
CHRM2 P08172 1/20 0.49
CHRM4 P08173 1/20 0.49
CHRM5 P08912 1/20 0.49
ADRA2A P08913 1/20 0.49
ADORA3 P0DMS8 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9479601 0.85 CYP2D6 (0.54) SIGMAR1CYP2C9CYP2C19CYP2D6ALDH1A1
SCHEMBL13664908 0.81 SIGMAR1 (0.56) SIGMAR1CYP2C9CYP2C19CYP2D6ALDH1A1
SCHEMBL4408727 0.77 SIGMAR1 (0.67) SIGMAR1CYP2C9CYP2C19CYP2D6ALDH1A1
SCHEMBL6339199 0.77 IDO1 (0.64) SIGMAR1CYP2C9CYP2C19CYP2D6ALDH1A1
SCHEMBL2743258 0.76 SIGMAR1 (0.67) SIGMAR1CYP2C9CYP2C19CYP2D6ALDH1A1
Hydrochloric Acid SCHEMBL7379764 0.76 SIGMAR1 (0.64) SIGMAR1CYP2C9CYP2C19CYP2D6ALDH1A1
SCHEMBL19041309 0.75 SIGMAR1 (0.58) SIGMAR1CYP2C9CYP2C19CYP2D6ALDH1A1
SCHEMBL29860963 0.75 SIGMAR1 (0.58) SIGMAR1CYP2C9CYP2C19CYP2D6ALDH1A1
SCHEMBL14112074 0.75 SIGMAR1 (0.50) SIGMAR1CYP2C9CYP2C19CYP2D6ALDH1A1
SCHEMBL13518880 0.75 SIGMAR1 (0.59) SIGMAR1CYP2C9CYP2C19CYP2D6ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1385514-A4 SPIROINDENE AND SPIROINDANE COMPOUNDS EURO CELTIQUE SA (LU) 2005-04-13 EP disclosed
EP-1385514-A1 SPIROINDENE AND SPIROINDANE COMPOUNDS Euro-Celtique S.A. (LU) 2004-02-04 EP disclosed
WO-2002085354-A1 SPIROINDENE AND SPIROINDANE COMPOUNDS EURO-CELTIQUE S.A. (LU) 2002-10-31 WO disclosed