SCHEMBL6169830

SCHEMBL6169830

CC(C)(C)OC(=O)N[C@@H](Cc1ccc(-c2cccc3ccccc23)cc1)C(=O)O

nearest known ligand 0.60

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 3/20 0.60
ACE P12821 3/20 0.57
CTSS P25774 5/20 0.56
CTSK P43235 4/20 0.56
PPARA Q07869 5/20 0.52
PPARG P37231 4/20 0.52
ITGB3 P05106 1/20 0.52
ITGA2B P08514 1/20 0.52
CTSB P07858 2/20 0.51
CTSL P07711 1/20 0.51
ITGA4 P13612 3/20 0.50
ITGB7 P26010 2/20 0.50
CYP2C9 P11712 1/20 0.50
CYP2C19 P33261 1/20 0.50
PPARD Q03181 1/20 0.50
MME P08473 1/20 0.50
ACE2 Q9BYF1 1/20 0.50
ITGB1 P05556 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1823733 0.90 CTSS (0.53) PTPN1ACECTSSCTSKPPARA
SCHEMBL8485076 0.89 CTSS (0.57) PTPN1ACECTSSCTSKPPARA
SCHEMBL1326276 0.86 CTSS (0.72) PTPN1ACECTSSCTSKPPARA
SCHEMBL1325181 0.86 CTSS (0.72) PTPN1ACECTSSCTSKPPARA
SCHEMBL1325182 0.86 CTSS (0.72) PTPN1ACECTSSCTSKPPARA
SCHEMBL23001196 0.86 PTPN1 (0.53) PTPN1ACECTSSCTSKPPARA
SCHEMBL13227703 0.85 PTPN1 (0.63) PTPN1ACECTSSCTSKPPARA
SCHEMBL3728073 0.84 PTPN1 (0.62) PTPN1ACECTSSCTSKPPARA
SCHEMBL3728076 0.84 PTPN1 (0.62) PTPN1ACECTSSCTSKPPARA
SCHEMBL3724246 0.83 ITGA4 (0.63) PTPN1ACEITGA4ITGB7ITGB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0888341-B1 NOVEL SULPHUR DERIVATIVES COMPRISING AN AMIDE BOND, METHOD FOR PREPARING SAME, USE THEREOF AS DRUGS, AND PHARMACEUTICAL COMPOSITIONS CONTAINING SUCH DERIVATIVES AVENTIS PHARMA SA (FR) 2005-11-30 EP disclosed
US-6136842-A INHIBITION OF ENDOTHELIN-CONVERTING ENZYME HOECHST MARION ROUSSEL (FR) 2000-10-24 US disclosed