SCHEMBL6170156

SCHEMBL6170156

Cc1ccnc(C(=O)c2[nH]c3cc(C(F)(F)F)ccc3c2C(C)C(=O)O)c1

nearest known ligand 0.50

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 9/20 0.50
PTGS1 P23219 7/20 0.50
KIF11 P52732 6/20 0.40
MAPT P10636 1/20 0.38
SORT1 Q99523 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6171485 0.92 PTGS2 (0.56) PTGS2PTGS1KIF11SORT1
SCHEMBL6172104 0.88 PTGS2 (0.53) PTGS2PTGS1
SCHEMBL6181624 0.87 PTGS2 (0.66) PTGS2PTGS1KIF11
SCHEMBL6171838 0.83 PTGS2 (0.67) PTGS2PTGS1KIF11
SCHEMBL6171712 0.83 PTGS2 (0.68) PTGS2PTGS1KIF11
SCHEMBL6171969 0.83 PTGS2 (0.67) PTGS2PTGS1MAPT
SCHEMBL6170712 0.82 PTGS2 (0.53) PTGS2PTGS1MAPT
SCHEMBL6171600 0.81 PTGS2 (0.58) PTGS2PTGS1MAPTSORT1
SCHEMBL6169979 0.81 PTGS2 (0.76) PTGS2PTGS1
SCHEMBL6173175 0.81 PTGS2 (0.69) PTGS2PTGS1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1045833-B1 2,3-SUBSTITUTED INDOLE COMPOUNDS AS COX-2 INHIBITORS PFIZER (US) 2005-11-02 EP claimed
US-6608070-B1 Useful for treatment of medical condition in which prostaglandins are implicated as pathogens NAKAO KAZUNARI (JP) 2003-08-19 US claimed
US-6608070-B1 Useful for treatment of medical condition in which prostaglandins are implicated as pathogens NAKAO KAZUNARI (JP) 2003-08-19 US disclosed