SCHEMBL6172992

SCHEMBL6172992

CC(C)(C)Oc1c(C#N)cccc1CBr

nearest known ligand 0.34

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 1/20 0.34
TSHR P16473 2/20 0.32
ALDH1A1 P00352 1/20 0.31
HTR1A P08908 1/20 0.31
ADRA2A P08913 1/20 0.31
ADRA2B P18089 1/20 0.31
MAOA P21397 1/20 0.31
HTR2B P41595 1/20 0.31
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
SSTR4 P31391 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7717027 0.81 TSHR (0.38) TSHRALDH1A1NPC1RAB9A
SCHEMBL1761160 0.78 DYRK1A (0.38) NAMPTTSHRALDH1A1HTR1AADRA2A
SCHEMBL4424952 0.75 AR (0.41) NAMPTTSHRALDH1A1NPC1RAB9A
SCHEMBL31667703 0.72 TSHR (0.43) TSHRALDH1A1
SCHEMBL6354890 0.72 TSHR (0.43) TSHRALDH1A1
SCHEMBL29513232 0.70 CYP19A1 (0.46) TSHRALDH1A1NPC1RAB9A
SCHEMBL899 0.70 CYP19A1 (0.46) TSHRALDH1A1NPC1RAB9A
SCHEMBL3053661 0.70 TSHR (0.35) TSHRALDH1A1NPC1RAB9A
SCHEMBL1232356 0.70 GABRA1 (0.37) TSHRALDH1A1
SCHEMBL1125092 0.70 SMN1; SMN2 (0.37) TSHRALDH1A1MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1254136-A4 FACTOR Xa INHIBITORS WITH ARYL-AMIDINES AND DERIVATIVES, AND PRODRUGS THEREOF LG CHEM INVESTMENT LTD (KR) 2005-06-01 EP disclosed
EP-1254136-A1 FACTOR Xa INHIBITORS WITH ARYL-AMIDINES AND DERIVATIVES, AND PRODRUGS THEREOF LG Chem Investment, Ltd. (KR) 2002-11-06 EP disclosed
WO-2001055146-A1 FACTOR Xa INHIBITORS WITH ARYL-AMIDINES AND DERIVATIVES, AND PRODRUGS THEREOF LG CHEM INVESTMENT LTD. (KR) 2001-08-02 WO disclosed