SCHEMBL6175754

SCHEMBL6175754

CC(c1cc(F)nc2ccccc12)C1NC(=O)N(c2ccc(SC(F)(F)F)cc2)C1=O

nearest known ligand 0.39

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.39
AR P10275 1/20 0.35
IGF1R P08069 9/20 0.34
TRPV4 Q9HBA0 1/20 0.33
PDE2A O00408 5/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6175824 0.91 LMNA (0.39) LMNAARIGF1RTRPV4PDE2A
SCHEMBL6172638 0.90 LMNA (0.39) LMNAARIGF1RTRPV4PDE2A
SCHEMBL6171605 0.90 LMNA (0.39) LMNAARIGF1RTRPV4PDE2A
SCHEMBL6175015 0.89 LMNA (0.38) LMNAARIGF1RTRPV4PDE2A
SCHEMBL6176997 0.86 KDM4E (0.42) LMNAARTRPV4PDE2A
SCHEMBL6174264 0.84 IGF1R (0.43) LMNAARIGF1R
SCHEMBL6173610 0.79 IGF1R (0.37) LMNAIGF1R
SCHEMBL6175139 0.79 LMNA (0.38) LMNAIGF1RTRPV4
SCHEMBL6171361 0.78 IGF1R (0.37) LMNAIGF1RTRPV4PDE2A
SCHEMBL6174667 0.77 LMNA (0.36) LMNAIGF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1599464-A2 NOVEL CYCLIC UREA DERIVATIVES, PREPARATION METHOD THEREOF AND PHARMACEUTICAL USE OF SAME AS KINASE INHIBITORS Aventis Pharma S.A. (FR) 2005-11-30 EP disclosed
WO-2004070050-A2 CYCLIC UREA DERIVATIVES, PREPARATION METHOD THEREOF AND PHARMACEUTICAL USE OF SAME AS KINASE INHIBITORS AVENTIS PHARMA S.A. (FR) 2004-08-19 WO disclosed