SCHEMBL6176019

SCHEMBL6176019

CCN(CC)CCN1C(=O)C(O)(c2ccccc2Cl)c2c1cc(C#CCCC(=O)NCCO)cc2C(F)(F)F

nearest known ligand 0.62

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GHSR Q92847 16/20 0.62
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
CHEK1 O14757 2/20 0.31
WEE1 P30291 2/20 0.31
CDK1 P06493 1/20 0.31
CCNB1 P14635 1/20 0.31
GAA P10253 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2581081 0.89 GHSR (0.65) GHSR
SCHEMBL2577500 0.88 GHSR (0.76) GHSR
SCHEMBL6177362 0.88 GHSR (0.80) GHSRMEN1KMT2A
SCHEMBL2577096 0.87 GHSR (0.66) GHSR
SCHEMBL2576235 0.86 GHSR (0.69) GHSR
SCHEMBL7842815 0.86 GHSR (0.75) GHSR
SCHEMBL2581006 0.85 GHSR (0.69) GHSR
SCHEMBL6179342 0.85 GHSR (0.66) GHSR
SCHEMBL6178087 0.84 GHSR (0.78) GHSRWEE1
SCHEMBL2578574 0.84 GHSR (0.66) GHSR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1105376-B1 OXINDOLE DERIVATIVES AS GROWTH HORMONE RELEASERS SUMITOMO PHARMA (JP) 2005-02-09 EP disclosed
US-6576656-B1 Such as 1-(2-diethylaminoethyl)-4-trifluoromethyl-6-carbamoyl-3-hydroxy-3-(2 -chlorophenyl)oxindole; growth hormone releaser SUMITOMO PHARMACEUTICALS CO., LTD. (JP) 2003-06-10 US disclosed