SCHEMBL6177883

SCHEMBL6177883

CCn1nc(-c2cccnc2)c(C(=O)COC)c(Nc2cccc(F)c2)c1=O.CCn1nc(-c2ccncc2)c(C(=O)CO)c(Nc2cccc(F)c2)c1=O

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 3/20 0.41
TBXAS1 P24557 1/20 0.39
CYP1A1 P04798 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP1B1 Q16678 1/20 0.37
ABL1 P00519 1/20 0.34
BCR P11274 1/20 0.34
TAAR1 Q96RJ0 1/20 0.34
CSNK1E P49674 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34
BUB1 O43683 2/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
ATR Q13535 1/20 0.33
ADORA3 P0DMS8 1/20 0.33
ADORA2A P29274 1/20 0.33
ADORA2B P29275 1/20 0.33
ADORA1 P30542 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3039618 0.94 TBXAS1 (0.44) PDE4BTBXAS1CYP1A1CYP1A2CYP1B1
SCHEMBL3033125 0.89 PDE4B (0.48) PDE4BCYP1A1CYP1A2CYP1B1BUB1
SCHEMBL1652540 0.83 PDE4B (0.56) PDE4BTBXAS1CYP1A1CYP1A2CYP1B1
SCHEMBL1653053 0.81 PDE4B (0.47) PDE4BCYP1A1CYP1A2CYP1B1BUB1
SCHEMBL4682246 0.81 PDE4B (0.47) PDE4BCYP1A1CYP1A2CYP1B1CSNK1E
SCHEMBL1653670 0.80 PDE4B (0.59) PDE4BCYP1A1CYP1A2CYP1B1BUB1
SCHEMBL4707336 0.77 PDE4B (0.56) PDE4B
SCHEMBL3033404 0.77 PDE4B (0.56) PDE4BTBXAS1TAAR1CSNK1EADORA3
SCHEMBL4052442 0.77 PDE4B (0.52) PDE4BTBXAS1TAAR1CSNK1E
SCHEMBL6174791 0.76 PDE4B (0.46) PDE4BTBXAS1CSNK1E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575926-A1 NEW PYRIDAZIN-3(2H)-ONE DERIVATIVES Almirall Prodesfarma, S.A. (ES) 2005-09-21 EP disclosed
WO-2004058729-A1 NEW PYRIDAZIN-3(2H)-ONE DERIVATIVES ALMIRALL PRODESFARMA SA (ES) 2004-07-15 WO disclosed