SCHEMBL6178245

SCHEMBL6178245

CCN(CC)CCCN1C(=O)C(O)(c2ccc3ccccc3c2)c2cc(Cl)ccc21

nearest known ligand 0.58

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GHSR Q92847 9/20 0.58
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
SCN9A Q15858 7/20 0.43
PIM1 P11309 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
TP53 P04637 2/20 0.40
MAPT P10636 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6179661 0.94 GHSR (0.65) GHSRMEN1KMT2ASCN9A
SCHEMBL6178800 0.82 GHSR (0.71) GHSRMEN1KMT2ASCN9ATP53
SCHEMBL6178715 0.82 GHSR (0.45) GHSRMEN1KMT2APIM1TDP1
SCHEMBL6178184 0.81 SCN9A (0.57) GHSRMEN1KMT2ASCN9APIM1
SCHEMBL6179600 0.80 GHSR (0.70) GHSRMEN1KMT2ASCN9A
SCHEMBL6180123 0.78 GHSR (0.69) GHSRMEN1KMT2ASCN9A
SCHEMBL7855737 0.77 GHSR (0.78) GHSRSCN9A
SCHEMBL6179529 0.76 GHSR (0.79) GHSRMEN1KMT2ASCN9A
SCHEMBL6177267 0.74 SCN9A (0.59) GHSRSCN9ATP53MAPT
SCHEMBL6177479 0.73 GHSR (1.00) GHSRMEN1KMT2ASCN9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1105376-B1 OXINDOLE DERIVATIVES AS GROWTH HORMONE RELEASERS SUMITOMO PHARMA (JP) 2005-02-09 EP disclosed
US-6576656-B1 Such as 1-(2-diethylaminoethyl)-4-trifluoromethyl-6-carbamoyl-3-hydroxy-3-(2 -chlorophenyl)oxindole; growth hormone releaser SUMITOMO PHARMACEUTICALS CO., LTD. (JP) 2003-06-10 US disclosed