SCHEMBL6179968

SCHEMBL6179968

Cc1cccc(CC(=O)c2ccc3nsnc3c2)n1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAPT P10636 7/20 0.46
LMNA P02545 1/20 0.46
NPC1 O15118 11/20 0.43
RAB9A P51151 10/20 0.43
MEN1 O00255 4/20 0.43
KMT2A Q03164 4/20 0.43
ALDH1A1 P00352 3/20 0.43
POLB P06746 1/20 0.43
HPGD P15428 1/20 0.43
MAPK1 P28482 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
SMN1; SMN2 Q16637 4/20 0.39
KDM4E B2RXH2 2/20 0.39
PDE10A Q9Y233 1/20 0.39
HTT P42858 1/20 0.38
GRM1 Q13255 1/20 0.38
GAA P10253 1/20 0.38
HSD17B10 Q99714 1/20 0.38
TGFBR1 P36897 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7184457 0.91 MAPT (0.40) MAPTLMNANPC1RAB9AMEN1
SCHEMBL6177854 0.83 NPC1 (0.57) MAPTNPC1RAB9AMEN1KMT2A
SCHEMBL6181864 0.76 MAPT (0.48) MAPTLMNANPC1RAB9AMEN1
SCHEMBL14592085 0.75 MEN1 (0.48) MAPTLMNANPC1RAB9AMEN1
SCHEMBL5199273 0.75 GRM5 (0.55) MAPTNPC1RAB9AMEN1KMT2A
SCHEMBL5695828 0.75 TGFBR1 (0.42) NPC1RAB9AKMT2AHPGDSMN1; SMN2
SCHEMBL4065212 0.75 HCAR3 (0.42) MAPTNPC1RAB9AMEN1KMT2A
SCHEMBL5200109 0.74 PIM1 (0.40) NPC1RAB9AMEN1KMT2AALDH1A1
SCHEMBL15069589 0.74 NPC1 (0.50) MAPTLMNANPC1RAB9AMEN1
SCHEMBL4032725 0.73 KDM4E (0.56) MAPTNPC1RAB9AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6906089-B2 Triarylimidazole derivatives as cytokine inhibitors SMITHKLINE BEECHAM CORPORATION (US) 2005-06-14 US disclosed
EP-1268465-B1 TRIARYLIMIDAZOLE DERIVATIVES AS CYTOKINE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2005-06-01 EP disclosed
US-20030149277-A1 Triarylimidazole derivatives as cytokine inhibitors SMITHKLINE BEECHAM CORPORATION 2003-08-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030149277-A1 Triarylimidazole derivatives as cytokine inhibitors IL2, IL2RA, IL6ST MAPT 4189/4885LMNA 3761/4885NPC1 1981/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.