SCHEMBL6180622

SCHEMBL6180622

CC(C)(C)N(C(=O)O)[C@H](C(=O)N1CCC[C@H]1C(=O)NC1CCc2n[nH]cc2C1)C(c1ccccc1)c1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SCN4A P35499 1/20 0.39
KCNH2 Q12809 1/20 0.37
KDM4E B2RXH2 1/20 0.37
MAPK1 P28482 1/20 0.37
CYP3A4 P08684 5/20 0.35
CYP2C9 P11712 5/20 0.35
CYP2C19 P33261 5/20 0.35
CYP1A2 P05177 2/20 0.35
CYP2D6 P10635 2/20 0.35
XIAP P98170 4/20 0.35
BIRC2 Q13490 8/20 0.34
BIRC3 Q13489 3/20 0.34
F2 P00734 1/20 0.34
ELANE P08246 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6178104 1.00 SCN4A (0.39) SCN4AKCNH2KDM4EMAPK1CYP3A4
SCHEMBL6179624 0.88 F2 (0.41) KCNH2F2
SCHEMBL6181452 0.85 XIAP (0.40) SCN4AXIAPF2
SCHEMBL6181742 0.85 KDM4E (0.41) SCN4AKCNH2KDM4EMAPK1CYP3A4
SCHEMBL6178057 0.85 KDM4E (0.41) SCN4AKCNH2KDM4EMAPK1CYP3A4
SCHEMBL6184253 0.84 SCN4A (0.41) SCN4AKCNH2KDM4EMAPK1CYP3A4
Hydrochloric Acid SCHEMBL6093429 0.84 KDM4E (0.40) SCN4AKCNH2KDM4EMAPK1CYP3A4
Hydrochloric Acid SCHEMBL6092133 0.84 KDM4E (0.40) SCN4AKCNH2KDM4EMAPK1CYP3A4
SCHEMBL6095258 0.83 KDM4E (0.39) SCN4AKCNH2KDM4EMAPK1CYP3A4
SCHEMBL6093041 0.83 KDM4E (0.39) SCN4AKCNH2KDM4EMAPK1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1287018-B1 THROMBIN INHIBITORS LEK TOVARNA FARMACEVTSKIH (SI) 2005-01-19 EP claimed