SCHEMBL6180652

SCHEMBL6180652

COc1ccccc1C1=CCN(CC(N)Cc2ccccc2)CC1

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PPARG P37231 1/20 0.52
PPARA Q07869 1/20 0.52
PARP1 P09874 1/20 0.46
HTR1A P08908 4/20 0.44
CCNT1 O60563 3/20 0.44
CDK9 P50750 3/20 0.44
CACNA1G O43497 1/20 0.43
KCNH2 Q12809 1/20 0.43
TNKS O95271 1/20 0.42
TNKS2 Q9H2K2 1/20 0.42
DRD2 P14416 2/20 0.41
SLC6A4 P31645 2/20 0.41
SLC6A3 Q01959 2/20 0.41
GNRHR P30968 2/20 0.41
KDM4E B2RXH2 1/20 0.40
MAPT P10636 1/20 0.40
HTR2A P28223 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8177719 0.83 SLC6A4 (0.39) PPARGPPARAHTR1ACCNT1CDK9
SCHEMBL8181908 0.83 SLC6A4 (0.39) PPARGPPARAHTR1ACCNT1CDK9
SCHEMBL2396688 0.82 HTR1A (0.57) PPARGPPARAPARP1HTR1ACCNT1
SCHEMBL6068434 0.81 TNKS (0.42) PPARGPPARAPARP1HTR1ACCNT1
Cyclohexane SCHEMBL6181993 0.79 PPARG (0.52) PPARGPPARAPARP1CCNT1CDK9
SCHEMBL6178407 0.77 CCNT1 (0.50) PPARGPPARACCNT1CDK9
SCHEMBL31348259 0.77 CCNT1 (0.52) PPARGPPARAPARP1HTR1ACCNT1
SCHEMBL31348196 0.77 CCNT1 (0.52) PPARGPPARAPARP1HTR1ACCNT1
SCHEMBL9278928 0.76 PPARG (0.53) PPARGPPARAPARP1HTR1ACCNT1
SCHEMBL6177022 0.76 MEN1 (0.51) PPARGPPARAHTR1ACCNT1CDK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140830-B1 ARYLPIPERIDINE AND ARYL-1,2,5,6-TETRAHYDROPYRIDINE AMIDE DERIVATIVES HAVING 5HT1A RECEPTOR ACTIVITY WYETH CORP (US) 2005-05-04 EP claimed
US-6503928-B2 Central nervous system disorders; psychological disorders WYETH 2003-01-07 US claimed
US-6503928-B2 Central nervous system disorders; psychological disorders WYETH 2003-01-07 US disclosed