SCHEMBL6181099

SCHEMBL6181099

CCCCCS(=O)(=O)NC(=O)c1ccc(N)c(N(C)Cc2ccc(Cl)cc2Cl)c1

nearest known ligand 0.54

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PPARG P37231 15/20 0.54
SCN9A Q15858 1/20 0.40
PTPN1 P18031 1/20 0.38
ALDH1A1 P00352 1/20 0.37
GAA P10253 1/20 0.37
HTT P42858 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6180762 0.86 PPARG (0.52) PPARGSCN9APTPN1ALDH1A1GAA
SCHEMBL6134825 0.81 PPARG (0.58) PPARGPTPN1
SCHEMBL6172090 0.78 PPARG (0.54) PPARG
SCHEMBL5881961 0.72 PPARG (0.54) PPARG
SCHEMBL6305809 0.72 PPARG (0.54) PPARGPTPN1
SCHEMBL6181103 0.72 THRB (0.40) PPARGALDH1A1GAAHTT
SCHEMBL5882208 0.72 PPARG (0.75) PPARG
SCHEMBL5881819 0.71 PPARG (0.62) PPARG
SCHEMBL5882012 0.71 PPARG (0.64) PPARG
SCHEMBL6299205 0.71 PPARG (0.55) PPARGPTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1000932-B9 AROMATIC RING DERIVATIVES FUJISAWA PHARMACEUTICAL CO (JP) 2005-12-28 EP disclosed
EP-1000932-B1 AROMATIC RING DERIVATIVES FUJISAWA PHARMACEUTICAL CO (JP) 2004-09-15 EP disclosed
US-6242474-B1 SULFONYLCARBAMOYLALKYLIMIDAZOLE DERIVATIVES; ANTIDIABETIC AGENTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-06-05 US disclosed
EP-1000932-A1 AROMATIC RING DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-05-17 EP disclosed