SCHEMBL6183448

SCHEMBL6183448

[CH2]Cc1ccc(Oc2cc(C#N)ccn2)cc1

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
P2RX3 P56373 9/20 0.45
FFAR1 O14842 1/20 0.43
LOXL2 Q9Y4K0 3/20 0.40
LOX P28300 1/20 0.39
ACACB O00763 1/20 0.38
OPRM1 P35372 1/20 0.38
GRM5 P41594 1/20 0.37
LMNA P02545 1/20 0.36
HTT P42858 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
GRIN1 Q05586 1/20 0.36
GRIN2B Q13224 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3163471 0.85 FFAR1 (0.46) P2RX3FFAR1LOXL2LOXACACB
SCHEMBL2145724 0.83 FFAR1 (0.47) P2RX3FFAR1LOXL2LOXOPRM1
SCHEMBL2427347 0.80 SMN1; SMN2 (0.46) P2RX3HTTSMN1; SMN2
SCHEMBL20239263 0.80 P2RX3 (0.44) P2RX3FFAR1LOXL2LOXACACB
SCHEMBL18049218 0.80 LOXL2 (0.53) P2RX3FFAR1LOXL2LOXACACB
SCHEMBL18249748 0.78 P2RX3 (0.47) P2RX3FFAR1LOXL2ACACBOPRM1
SCHEMBL20239266 0.76 FFAR1 (0.52) P2RX3FFAR1LOXL2ACACBOPRM1
SCHEMBL28895924 0.74 P2RX3 (0.41) P2RX3FFAR1LOXL2
SCHEMBL3158059 0.73 LOXL2 (0.44) P2RX3FFAR1LOXL2LOXACACB
SCHEMBL3173384 0.73 MAP4K4 (0.42) P2RX3FFAR1LOXL2LOXACACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1562595-A1 DIARYL ETHERS AS OPIOID RECEPTOR ANTAGONISTS ELI LILLY AND COMPANY (US) 2005-08-17 EP disclosed
WO-2004026305-A1 DIARYL ETHERS AS OPIOID RECEPTOR ANTAGONIST ELI LILLY AND COMPANY (US) 2004-04-01 WO disclosed