SCHEMBL6183696

SCHEMBL6183696

COc1ccc(OC)c(C(C(N)=O)c2ccccc2)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 3/20 0.50
ADRA2A P08913 2/20 0.50
KMT2A Q03164 4/20 0.49
MEN1 O00255 3/20 0.49
CYP2D6 P10635 1/20 0.49
LMNA P02545 3/20 0.48
ALDH1A1 P00352 2/20 0.48
MAPT P10636 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
MAPK1 P28482 1/20 0.48
BLM P54132 1/20 0.48
CYP1A2 P05177 1/20 0.46
TSHR P16473 1/20 0.46
CYP2C19 P33261 1/20 0.46
ADORA3 P0DMS8 1/20 0.46
HTT P42858 1/20 0.45
EPHX1 P07099 1/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7815176 0.91 ADRA1A (0.53) ADRA1AADRA2AKMT2AMEN1CYP2D6
SCHEMBL4504292 0.85 IDO1 (0.51) KMT2AMEN1LMNAALDH1A1MAPT
SCHEMBL17414457 0.81 KLK7 (0.55) KMT2AMEN1LMNAALDH1A1MAPT
SCHEMBL4493891 0.80 ACP3 (0.57) KMT2AMEN1ALDH1A1MAPTNPSR1
SCHEMBL30943709 0.77 ADRA2A (0.57) ADRA1AADRA2AKMT2AMEN1CYP2D6
SCHEMBL8806213 0.77 ADRA2A (0.57) ADRA1AADRA2AKMT2AMEN1CYP2D6
SCHEMBL15643615 0.76 KMT2A (0.52) KMT2AMEN1LMNAALDH1A1MAPT
SCHEMBL6755543 0.75 KMT2A (0.50) KMT2AMEN1LMNAALDH1A1MAPT
SCHEMBL4670011 0.75 CYP2D6 (0.56) ADRA1AADRA2AKMT2AMEN1CYP2D6
SCHEMBL23414454 0.74 ADRA1A (0.59) ADRA1AADRA2AKMT2AMEN1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1562919-A1 PHENYLALKYL AND PYRIDYLALKYL PIPERAZINE DERIVATIVES Warner-Lambert Company LLC (US) 2005-08-17 EP disclosed
WO-2004041793-A1 PHENYLALKYL AND PYRIDYLALKYL PIPERAZINE DERIVATIVES WARNER-LAMBERT COMPANY LLC (US) 2004-05-21 WO disclosed