SCHEMBL6184598

SCHEMBL6184598

N#Cc1cc(CCC(=O)O)ccc1N

nearest known ligand 0.49

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 14/20 0.49
FFAR4 Q5NUL3 4/20 0.48
AKR1B1 P15121 1/20 0.43
KEAP1 Q14145 1/20 0.43
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
SLC22A12 Q96S37 1/20 0.42
S1PR1 P21453 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1932268 0.87 FFAR1 (0.52) FFAR1FFAR4AKR1B1KEAP1CA1
SCHEMBL4030930 0.82 CHEK1 (0.42) FFAR1FFAR4S1PR1
SCHEMBL4022687 0.82 RAB9A (0.46)
SCHEMBL4715830 0.81 S1PR1 (0.58) FFAR1FFAR4AKR1B1KEAP1SLC22A12
SCHEMBL31230431 0.80 KDM4E (0.42) CA1CA2
SCHEMBL11685559 0.80 KDM4E (0.42) CA1CA2
SCHEMBL1002974 0.79 FFAR1 (0.53) FFAR1FFAR4KEAP1CA1CA2
SCHEMBL3352567 0.79 FFAR1 (0.53) FFAR1FFAR4AKR1B1KEAP1CA1
SCHEMBL23077756 0.78 CYP1A2 (0.49) FFAR1FFAR4S1PR1
SCHEMBL8385915 0.78 MAOB (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1537075-A2 DIARYLUREA DERIVATIVES AND THEIR USE AS CHLORIDE CHANNEL BLOCKERS NEUROSEARCH A/S (DK) 2005-06-08 EP disclosed
WO-2004022529-A2 DIARYLUREA DERIVATIVES AND THEIR USE AS CHLORIDE CHANNEL BLOCKERS NEUROSEARCH A/S (DK) 2004-03-18 WO disclosed