SCHEMBL6184752

SCHEMBL6184752

COc1c(OCC2CCN(C)CC2)ccc2c(Nc3ccc(Oc4cccnc4)cc3)c(C#N)cnc12

nearest known ligand 0.52

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 7/20 0.52
SRC P12931 7/20 0.52
ABL2 P42684 7/20 0.52
EGFR P00533 6/20 0.46
MAP2K1 Q02750 7/20 0.46
RAF1 P04049 5/20 0.46
MAPK3 P27361 1/20 0.44
MAPK1 P28482 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6182185 0.85 ABL1 (0.69) ABL1SRCABL2EGFRMAP2K1
SCHEMBL7002867 0.84 MAP2K1 (0.64) SRCMAP2K1RAF1MAPK3MAPK1
SCHEMBL6188532 0.79 SRC (0.73) ABL1SRCABL2
SCHEMBL6183868 0.79 SRC (0.74) ABL1SRCABL2
SCHEMBL6382824 0.78 MAP2K1 (0.68) SRCEGFRMAP2K1RAF1MAPK3
SCHEMBL7001258 0.77 MAP2K1 (0.57) MAP2K1RAF1MAPK3MAPK1
SCHEMBL6184215 0.77 SRC (0.73) ABL1SRCABL2
SCHEMBL6183312 0.77 SRC (0.73) ABL1SRCABL2EGFR
SCHEMBL6183229 0.76 MAP2K1 (0.57) SRCMAP2K1RAF1MAPK3MAPK1
SCHEMBL28909732 0.76 EGFR (0.70) EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1499594-B1 PROCESS FOR THE PREPARATION OF 7-SUBSTITUTED-3-QUINOLINE AND 3-QUINOL-4-ONE CARBONITRILES WYETH CORP (US) 2005-08-17 EP claimed