SCHEMBL6185985

SCHEMBL6185985

CC(=O)N(Cl)c1ccc(C)cc1.O=C(CCl)NC1c2ccccc2CC1O

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MMP9 P14780 10/20 0.43
MMP2 P08253 8/20 0.43
MMP1 P03956 7/20 0.43
MMP8 P22894 6/20 0.43
VIPR2 P41587 1/20 0.41
ALDH1A1 P00352 2/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
PSEN1 P49768 1/20 0.39
PSEN2 P49810 1/20 0.39
APH1B Q8WW43 1/20 0.39
NCSTN Q92542 1/20 0.39
APH1A Q96BI3 1/20 0.39
PSENEN Q9NZ42 1/20 0.39
MTNR1A P48039 1/20 0.38
MTNR1B P49286 1/20 0.38
ADAMTS4 O75173 1/20 0.38
ADAMTS5 Q9UNA0 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1273790 0.83 MMP9 (0.53) MMP9MMP2MMP1MMP8ALDH1A1
SCHEMBL1177439 0.83 MMP9 (0.53) MMP9MMP2MMP1MMP8ALDH1A1
SCHEMBL4858952 0.83 MMP9 (0.53) MMP9MMP2MMP1MMP8ALDH1A1
SCHEMBL8090956 0.83 MMP9 (0.53) MMP9MMP2MMP1MMP8ALDH1A1
SCHEMBL23343881 0.73 MMP9 (0.56) MMP9MMP2MMP1MMP8ALDH1A1
SCHEMBL14224779 0.73 MMP9 (0.56) MMP9MMP2MMP1MMP8ALDH1A1
SCHEMBL6186455 0.73 MMP1 (0.38) MMP9MMP2MMP1MMP8ALDH1A1
SCHEMBL2442157 0.71 MEN1 (0.54) MMP9MMP2MMP1MMP8ALDH1A1
SCHEMBL7740807 0.71 MEN1 (0.54) MMP9MMP2MMP1MMP8ALDH1A1
SCHEMBL885306 0.71 MEN1 (0.54) MMP9MMP2MMP1MMP8ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1567525-A2 SUBSTITUTED PIPERAZINE COMPOUNDS AND THEIR USE AS FATTY ACID OXIDATION INHIBITORS CV THERAPEUTICS, INC. (US) 2005-08-31 EP disclosed
WO-2004052887-A2 SUBSTITUTED PIPERAZINE COMPOUNDS AND THEIR USE AS FATTY ACID OXIDATION INHIBITORS CV THERAPEUTICS, INC. (US) 2004-06-24 WO disclosed