SCHEMBL6188099

SCHEMBL6188099

Fc1cc(F)cc(-c2[c]nccc2)c1

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.37
GRM5 P41594 1/20 0.35
NISCH Q9Y2I1 1/20 0.32
ATP1A1 P05023 1/20 0.31
ATP1B1 P05026 1/20 0.31
ATP1A3 P13637 1/20 0.31
ATP1B2 P14415 1/20 0.31
ATP1A2 P50993 1/20 0.31
ATP1B3 P54709 1/20 0.31
FXYD2 P54710 1/20 0.31
ATP1A4 Q13733 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5318660 0.85 NISCH (0.41) NOTUMGRM5NISCH
SCHEMBL4590846 0.82 MAPK14 (0.35)
SCHEMBL4909130 0.75
SCHEMBL19439 0.74 NOTUM (0.39) NOTUMNISCH
SCHEMBL5121103 0.73 NISCH (0.43) NISCH
SCHEMBL5543084 0.73 KMO (0.38)
SCHEMBL5797199 0.72 MAPT (0.43) NOTUM
SCHEMBL10561624 0.72 CYP3A4 (0.33)
SCHEMBL2412002 0.69 NOTUM (0.39) NOTUM
SCHEMBL4489657 0.69 CYP2A6 (0.56)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1585727-A1 INDOLES USEFUL IN THE TREATMENT OF ANDROGEN-RECEPTOR RELATED DISEASES Akzo Nobel N.V. (NL) 2005-10-19 EP disclosed
WO-2004041782-A1 INDOLES USEFUL IN THE TREATMENT OF ANDROGEN-RECEPTOR RELATED DISEASES AKZO NOBEL N.V. (NL) 2004-05-21 WO disclosed