SCHEMBL6188306

SCHEMBL6188306

CON(C)C(=O)c1cc(OCC(C)C)ccc1N

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
XDH P47989 2/20 0.44
SIRT2 Q8IXJ6 1/20 0.42
MAPT P10636 4/20 0.41
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 2/20 0.41
NPSR1 Q6W5P4 1/20 0.41
RXFP1 Q9HBX9 1/20 0.41
ABL1 P00519 1/20 0.41
CLK1 P49759 1/20 0.39
DYRK1A Q13627 1/20 0.39
DYRK1B Q9Y463 1/20 0.39
TP53 P04637 2/20 0.38
GAA P10253 2/20 0.38
NPC1 O15118 1/20 0.38
HTT P42858 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
NOS2 P35228 1/20 0.37
FOS P01100 1/20 0.37
JUN P05412 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3469683 0.83 CLK1 (0.55) MAPTKDM4EALDH1A1NPSR1CLK1
SCHEMBL1795616 0.82 KDM4E (0.55) XDHSIRT2MAPTKDM4EALDH1A1
SCHEMBL8136810 0.81 ALDH1A1 (0.47) XDHSIRT2MAPTKDM4EALDH1A1
SCHEMBL8206423 0.80 CYP1A2 (0.49) XDHSIRT2MAPTKDM4EALDH1A1
SCHEMBL6187334 0.78 FFAR1 (0.46) SIRT2TSHR
SCHEMBL12165513 0.75 MAPT (0.46) MAPTKDM4EALDH1A1CLK1DYRK1A
SCHEMBL26732 0.74 ABL1 (0.49) KDM4EALDH1A1ABL1CLK1DYRK1A
SCHEMBL28132 0.74 KDM4E (0.54) MAPTKDM4EALDH1A1CLK1DYRK1A
SCHEMBL2472646 0.74 KEAP1 (0.54) MAPTKDM4EALDH1A1CLK1DYRK1A
SCHEMBL3890176 0.74 CA12 (0.41) MAPTKDM4EALDH1A1CLK1DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0979227-B1 4,1-BENZOXAZEPINES, THEIR ANALOGUES, AND THEIR USE AS SOMATOSTATIN AGONISTS TAKEDA PHARMACEUTICAL (JP) 2005-11-16 EP disclosed
US-6352982-B1 TREATING DIABETES, OBESITY, OR INVETERATE DIARRHEA IN A MAMMAL WHICH COMPRISES ADMINISTERING AN EFFECTIVE AMOUNT OF A COMPOUND OF TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-03-05 US disclosed