SCHEMBL6188434

SCHEMBL6188434

COC(N)Cc1ccc(-c2ccccc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRR Q9GZT4 2/20 0.49
PSAT1 Q9Y617 2/20 0.49
EPHX1 P07099 1/20 0.48
IDO1 P14902 2/20 0.47
AGXT P21549 2/20 0.47
TAAR1 Q96RJ0 4/20 0.47
PPARG P37231 7/20 0.47
PPARA Q07869 6/20 0.47
PPARD Q03181 1/20 0.47
SLC6A2 P23975 2/20 0.45
MAOA P21397 1/20 0.45
SLC6A4 P31645 1/20 0.45
SLC6A3 Q01959 1/20 0.45
SIGMAR1 Q99720 1/20 0.45
CYP2A6 P11509 1/20 0.45
ADORA2A P29274 1/20 0.45
ADORA1 P30542 1/20 0.45
MMP12 P39900 1/20 0.44
CYP2D6 P10635 2/20 0.43
CYP1A2 P05177 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL479459 0.88 EPHX1 (0.62) EPHX1TAAR1SLC6A2MAOASLC6A4
SCHEMBL4950704 0.88 EPHX1 (0.62) EPHX1TAAR1SLC6A2MAOASLC6A4
SCHEMBL4950924 0.88 EPHX1 (0.62) EPHX1TAAR1SLC6A2MAOASLC6A4
Hydrochloric Acid SCHEMBL28001158 0.86 EPHX1 (0.60) SRREPHX1TAAR1SLC6A2MAOA
Iodide SCHEMBL28946993 0.86 EPHX1 (0.60) EPHX1TAAR1SLC6A2MAOASLC6A4
SCHEMBL17413364 0.78 TAAR1 (0.75) TAAR1SLC6A2MAOASLC6A4SLC6A3
SCHEMBL9417738 0.78 TAAR1 (0.75) TAAR1SLC6A2MAOASLC6A4SLC6A3
SCHEMBL16389766 0.78 SLC6A4 (0.44) EPHX1TAAR1SLC6A4CYP2D6CYP1A2
SCHEMBL4075991 0.78 TAAR1 (0.75) TAAR1SLC6A2MAOASLC6A4SLC6A3
SCHEMBL22861986 0.77 TAAR1 (0.56) SRRPSAT1EPHX1IDO1AGXT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1542977-A1 2,5-DIOXOIMIDAZOLIDIN-4-YL ACETAMIDES AND ANALOGUES AS INHIBITORS OF METALLOPROTEINASE MMP12. AstraZeneca AB (SE) 2005-06-22 EP disclosed
WO-2004020415-A1 2,5-DIOXOIMIDAZOLIDIN-4-YL ACETAMIDES AND ANALOGUES AS INHIBITORS OF METALLOPROTEINASE MMP12. ASTRAZENECA AB (SE) 2004-03-11 WO disclosed