SCHEMBL6188508

SCHEMBL6188508

COc1cccc(OC)c1C(=O)c1c(C)[nH]c2ccc(NC(=O)C3CCCCC3)cc12

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.51
MAOB P27338 1/20 0.51
POLB P06746 1/20 0.48
SMN1; SMN2 Q16637 2/20 0.47
GRM4 Q14833 1/20 0.47
ULK1 O75385 1/20 0.47
ITK Q08881 3/20 0.47
NPSR1 Q6W5P4 1/20 0.46
MTNR1A P48039 1/20 0.46
MTNR1B P49286 1/20 0.46
STK17B O94768 1/20 0.46
STK17A Q9UEE5 1/20 0.46
ALDH1A1 P00352 2/20 0.45
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
KDM4E B2RXH2 1/20 0.43
NPC1 O15118 1/20 0.43
CYP1A2 P05177 1/20 0.43
PKM P14618 1/20 0.43
HPGD P15428 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6185392 0.99 MAOA (0.49) MAOAMAOBPOLBSMN1; SMN2GRM4
SCHEMBL6187015 0.97 ULK1 (0.49) MAOAMAOBPOLBSMN1; SMN2GRM4
SCHEMBL6188504 0.89 GRM4 (0.51) MAOAMAOBPOLBSMN1; SMN2GRM4
SCHEMBL6188606 0.88 MAOA (0.55) MAOAMAOBSMN1; SMN2ITKNPSR1
SCHEMBL6185134 0.87 MAOA (0.54) MAOAMAOBSMN1; SMN2GRM4ITK
SCHEMBL6189495 0.87 PARP1 (0.45) MAOAMAOBPOLBULK1MTNR1A
SCHEMBL6189454 0.87 MAOA (0.53) MAOAMAOBPOLBSMN1; SMN2ULK1
SCHEMBL6189592 0.85 MAOA (0.51) MAOAMAOBPOLBSMN1; SMN2ULK1
SCHEMBL6187132 0.85 MAOA (0.50) MAOAMAOBPOLBSMN1; SMN2ULK1
SCHEMBL6186285 0.84 MAOA (0.49) MAOAMAOBPOLBSMN1; SMN2ULK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1554271-A1 SUBSTITUTED INDOLES AND THEIR USE AS HCV INHIBITORS Rigel Pharmaceuticals, Inc. (US) 2005-07-20 EP disclosed
WO-2004035571-A1 SUBSTITUTED INDOLES AND THEIR USE AS HCV INHIBITORS RIGEL PHARMACEUTICALS, INC. (US) 2004-04-29 WO disclosed