SCHEMBL6193458

SCHEMBL6193458

Cc1cccc(C(N)=O)c1Nc1nc(Cl)ncc1[N+](=O)[O-]

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 6/20 0.54
MAPT P10636 4/20 0.48
NPC1 O15118 2/20 0.48
ALDH1A1 P00352 2/20 0.48
RAB9A P51151 2/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
JAK3 P52333 6/20 0.44
TYK2 P29597 5/20 0.44
JAK2 O60674 3/20 0.44
LCK P06239 2/20 0.44
PTK2B Q14289 2/20 0.44
GSK3B P49841 2/20 0.44
CDC7 O00311 1/20 0.44
PLK4 O00444 1/20 0.44
CHEK1 O14757 1/20 0.44
DCLK1 O15075 1/20 0.44
CHUK O15111 1/20 0.44
PDPK1 O15530 1/20 0.44
DAPK3 O43293 1/20 0.44
DYRK3 O43781 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1080985 0.84 JAK3 (0.47) ALDH1A1RAB9ASMN1; SMN2JAK3TYK2
SCHEMBL1204172 0.82 PIN1 (0.62) PIN1SMN1; SMN2JAK3TYK2JAK2
SCHEMBL29549327 0.77 PIN1 (0.51) PIN1MAPTALDH1A1SMN1; SMN2LCK
SCHEMBL22807430 0.77 PIN1 (0.51) PIN1MAPTALDH1A1SMN1; SMN2LCK
SCHEMBL3811000 0.77 PIN1 (0.58) PIN1MAPTJAK3TYK2JAK2
SCHEMBL3807303 0.75 PIN1 (0.53) PIN1MAPTJAK3TYK2JAK2
SCHEMBL8298042 0.75 PIN1 (0.58) PIN1MAPTALDH1A1PTK2BGSK3B
SCHEMBL3814860 0.75 PIN1 (0.62) PIN1MAPTJAK3TYK2JAK2
SCHEMBL6193447 0.75 PRKCQ (0.53) PIN1GSK3BDCLK1PRKD3MAP4K4
SCHEMBL16012501 0.75 PIN1 (0.68) PIN1MAPTSMN1; SMN2JAK2PTK2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1597251-A2 PYRIMIDINE COMPOUNDS SmithKline Beecham Corporation (US) 2005-11-23 EP disclosed
WO-2004074244-A2 PYRIMIDINE COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2004-09-02 WO disclosed