SCHEMBL6196703

SCHEMBL6196703

COC(=O)COCC1=CNC(=O)N(C(=O)Oc2ccc([N+](=O)[O-])cc2)C1c1ccc(F)c(F)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.36
ADRA1D P25100 2/20 0.35
ADRA1A P35348 2/20 0.35
ADRA1B P35368 2/20 0.35
BCL9 O00512 1/20 0.33
CTNNB1 P35222 1/20 0.33
KDM1A O60341 1/20 0.33
ALDH1A1 P00352 2/20 0.33
GAA P10253 2/20 0.33
THRB P10828 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C19 P33261 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
CACNA1F O60840 1/20 0.33
CACNA1D Q01668 1/20 0.33
CACNA1S Q13698 1/20 0.33
CACNA1C Q13936 1/20 0.33
KMT2A Q03164 1/20 0.32
MGLL Q99685 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6196706 0.79 ADRA1D (0.34) ADRA1DADRA1AADRA1BKDM1ACACNA1F
SCHEMBL6198367 0.78 ADRA1D (0.41) ADRA1DADRA1AADRA1BALDH1A1RAB9A
SCHEMBL6196834 0.76 ADRA1D (0.51) ADRA1DADRA1AADRA1B
SCHEMBL6198625 0.76 ADRA1D (0.45) ADRA1DADRA1AADRA1BCACNA1FCACNA1D
SCHEMBL7674379 0.76 ADRA1D (0.51) ADRA1DADRA1AADRA1B
SCHEMBL6715316 0.76 CACNA1F (0.44) ADRA1DADRA1AADRA1BCACNA1FCACNA1D
SCHEMBL6193641 0.75 ADRA1D (0.54) ADRA1DADRA1AADRA1BCACNA1FCACNA1D
SCHEMBL7162576 0.75 ADRA1D (0.54) ADRA1DADRA1AADRA1BCACNA1FCACNA1D
SCHEMBL6715576 0.73 CACNA1F (0.48) ADRA1DADRA1AADRA1BCACNA1FCACNA1D
SCHEMBL6772155 0.73 CACNA1F (0.39) ADRA1DADRA1AADRA1BALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1021185-A4 DIDHYDROPYRIMIDINES AND USES THEREOF SYNAPTIC PHARMA CORP (US) 2005-09-07 EP disclosed
EP-1021185-A1 DIDHYDROPYRIMIDINES AND USES THEREOF SYNAPTIC PHARMACEUTICAL CORPORATION (US) 2000-07-26 EP disclosed
WO-1997042956-A1 DIDHYDROPYRIMIDINES AND USES THEREOF SYNAPTIC PHARMACEUTICAL CORPORATION (US) 1997-11-20 WO disclosed