SCHEMBL6199790

SCHEMBL6199790

CCOC(=O)C1=C(C)N=C(SCc2ccc(OC)cc2)NC1c1ccc([N+](=O)[O-])cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.47
SMN1; SMN2 Q16637 4/20 0.47
MAPT P10636 1/20 0.47
ADORA3 P0DMS8 1/20 0.46
HTT P42858 4/20 0.44
LMNA P02545 4/20 0.44
CRHBP P24387 1/20 0.44
CRHR2 Q13324 1/20 0.44
GAA P10253 2/20 0.44
POLB P06746 2/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
NCOA1 Q15788 1/20 0.43
NCOA3 Q9Y6Q9 1/20 0.43
TSHR P16473 1/20 0.43
KDR P35968 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6201423 0.93 MAPT (0.48) ALDH1A1SMN1; SMN2MAPTADORA3HTT
SCHEMBL6201427 0.76 ALDH1A1 (0.43) ALDH1A1SMN1; SMN2MAPTHTTLMNA
SCHEMBL27875502 0.76 SMN1; SMN2 (0.52) ALDH1A1SMN1; SMN2MAPTADORA3LMNA
SCHEMBL28024258 0.75 ALDH1A1 (0.55) ALDH1A1SMN1; SMN2MAPTHTTLMNA
SCHEMBL9476034 0.72 ALDH1A1 (0.49) ALDH1A1SMN1; SMN2MAPTHTTLMNA
SCHEMBL9475602 0.72 MAPT (0.49) ALDH1A1SMN1; SMN2MAPTHTTLMNA
SCHEMBL10911202 0.71 POLB (0.40) ALDH1A1SMN1; SMN2MAPTLMNAGAA
SCHEMBL10736837 0.71 ALDH1A1 (0.45) ALDH1A1SMN1; SMN2MAPTHTTMEN1
SCHEMBL10826912 0.71 CACNA1C (0.54) HTTGAAMEN1KMT2ATSHR
SCHEMBL6194820 0.71 MAPT (0.47) ALDH1A1SMN1; SMN2MAPTHTTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1021185-A4 DIDHYDROPYRIMIDINES AND USES THEREOF SYNAPTIC PHARMA CORP (US) 2005-09-07 EP disclosed
EP-1021185-A1 DIDHYDROPYRIMIDINES AND USES THEREOF SYNAPTIC PHARMACEUTICAL CORPORATION (US) 2000-07-26 EP disclosed
WO-1997042956-A1 DIDHYDROPYRIMIDINES AND USES THEREOF SYNAPTIC PHARMACEUTICAL CORPORATION (US) 1997-11-20 WO disclosed