SCHEMBL6199828

SCHEMBL6199828

COc1cc2c(cc1O)CCC2=O.COc1cc2c(cc1OC)C(=O)CC2

nearest known ligand 0.87

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.56
ACHE P22303 3/20 0.54
MAOA P21397 3/20 0.53
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
CHRNA7 P36544 1/20 0.45
KDM4E B2RXH2 1/20 0.45
ALDH1A1 P00352 1/20 0.45
HSD17B1 P14061 1/20 0.44
CYP3A4 P08684 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3081446 0.97 PTGS2 (0.59) PTGS2ACHEMAOACHRNA7KDM4E
SCHEMBL662848 0.93 ACHE (0.57) PTGS2ACHEMAOACHRNA7
SCHEMBL354177 0.89 KMT2A (0.56) ACHEMAOAMEN1KMT2AKDM4E
SCHEMBL29420326 0.89 KMT2A (0.56) ACHEMAOAMEN1KMT2AKDM4E
SCHEMBL29420327 0.89 KMT2A (0.56) ACHEMAOAMEN1KMT2AKDM4E
SCHEMBL6214359 0.89 PTGS2 (0.47) PTGS2ACHEMAOAMEN1KMT2A
SCHEMBL1274990 0.87 ACHE (0.54) PTGS2ACHEMAOAMEN1KMT2A
SCHEMBL1545375 0.87 ACHE (0.54) PTGS2ACHEMAOAMEN1KMT2A
SCHEMBL9620643 0.83 ACHE (0.54) PTGS2ACHEMAOACHRNA7HSD17B1
SCHEMBL661560 0.83 ACHE (0.54) PTGS2ACHEMAOAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1603885-A1 FUSED TRI AND TETRA-CYCLIC PYRAZOLE KINASE INHIBITORS Abbott Laboratories (US) 2005-12-14 EP disclosed
WO-2004080973-A1 FUSED TRI AND TETRA-CYCLIC PYRAZOLE KINASE INHIBITORS ABBOTT LABORATORIES (US) 2004-09-23 WO disclosed