SCHEMBL6200702

SCHEMBL6200702

O=C(O)c1c(CN2CCC(O)C2)c(-c2ccccc2)nc2ccccc12

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TACR2 P21452 14/20 0.51
TACR3 P29371 13/20 0.51
OPRM1 P35372 6/20 0.51
TRPV4 Q9HBA0 2/20 0.50
PDE10A Q9Y233 2/20 0.49
LMNA P02545 2/20 0.49
DHODH Q02127 2/20 0.49
TSHR P16473 1/20 0.48
POLB P06746 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6202262 1.00 TACR2 (0.51) TACR2TACR3OPRM1TRPV4PDE10A
SCHEMBL6200694 1.00 TACR2 (0.51) TACR2TACR3OPRM1TRPV4PDE10A
SCHEMBL5733751 0.87 TACR3 (0.62) TACR2TACR3OPRM1TRPV4
SCHEMBL5945331 0.85 TACR2 (0.67) TACR2TACR3OPRM1TRPV4PDE10A
SCHEMBL6852921 0.84 TACR2 (0.53) TACR2TACR3OPRM1TRPV4PDE10A
SCHEMBL6857830 0.83 TACR2 (0.55) TACR2TACR3OPRM1TRPV4PDE10A
Hydrochloric Acid SCHEMBL6851636 0.83 TACR3 (0.52) TACR2TACR3OPRM1TRPV4
SCHEMBL5635546 0.82 TACR3 (0.76) TACR2TACR3OPRM1TRPV4
SCHEMBL8116231 0.82 TACR3 (0.76) TACR2TACR3OPRM1TRPV4
SCHEMBL6848843 0.82 TACR3 (0.58) TACR2TACR3OPRM1TRPV4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1377567-B1 QUINOLINE-4-CARBOXAMIDE DERIVATIVES AS NK-3 AND NK-2 RECEPTOR ANTAGONISTS GLAXOSMITHKLINE SPA (IT) 2005-12-21 EP claimed