SCHEMBL6848843

SCHEMBL6848843

O=C(O)c1c(CN2CCN3CCCC3C2)c(-c2ccccc2)nc2ccccc12

nearest known ligand 0.58

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 12/20 0.58
TACR2 P21452 10/20 0.58
OPRM1 P35372 5/20 0.58
KCNH2 Q12809 3/20 0.56
TRPV4 Q9HBA0 8/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6855974 0.90 TACR3 (0.70) TACR3TACR2OPRM1KCNH2TRPV4
SCHEMBL2373330 0.85 TRPV4 (0.72) TACR3TACR2OPRM1KCNH2TRPV4
Hydrochloric Acid SCHEMBL5733490 0.84 TRPV4 (0.71) TACR3TACR2OPRM1KCNH2TRPV4
SCHEMBL6853726 0.84 TACR3 (0.60) TACR3TACR2OPRM1KCNH2TRPV4
SCHEMBL4236971 0.82 TACR3 (0.85) TACR3TACR2KCNH2
SCHEMBL6200694 0.82 TACR2 (0.51) TACR3TACR2OPRM1TRPV4
SCHEMBL6200702 0.82 TACR2 (0.51) TACR3TACR2OPRM1TRPV4
SCHEMBL6202262 0.82 TACR2 (0.51) TACR3TACR2OPRM1TRPV4
SCHEMBL6853853 0.82 TRPV4 (0.62) TACR3TACR2OPRM1KCNH2TRPV4
SCHEMBL5733751 0.80 TACR3 (0.62) TACR3TACR2OPRM1KCNH2TRPV4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6780875-B2 RESPIRATORY SYSTEM DISORDERS; ANTIINFLAMMATORY AGENTS; PSYCHOLOGICAL DISORDERS SMITHKLINE BEECHAM S.P.A. (IT) 2004-08-24 US claimed
US-6780875-B2 RESPIRATORY SYSTEM DISORDERS; ANTIINFLAMMATORY AGENTS; PSYCHOLOGICAL DISORDERS SMITHKLINE BEECHAM S.P.A. (IT) 2004-08-24 US disclosed