SCHEMBL6201771

SCHEMBL6201771

Nc1cc(N)c2[nH]c(=O)[nH]c(=O)c2c1

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 8/20 0.39
GDA Q9Y2T3 1/20 0.37
KDM4E B2RXH2 2/20 0.35
CA12 O43570 2/20 0.35
CA9 Q16790 2/20 0.35
TYMP P19971 5/20 0.34
GSK3B P49841 1/20 0.34
BACE1 P56817 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HPGD P15428 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
XDH P47989 1/20 0.33
PNP P00491 1/20 0.33
MAPT P10636 1/20 0.33
TYMS P04818 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20853010 0.81 TYMP (0.39) PARP1GDAKDM4ECA12CA9
SCHEMBL5357075 0.75 SIRT2 (0.44) PARP1KDM4ECA12CA9ALDH1A1
SCHEMBL2267356 0.75 CHUK (0.36) PARP1ALDH1A1
SCHEMBL6199860 0.72 PARP1 (0.67) PARP1KDM4ECA12CA9ALDH1A1
SCHEMBL4610600 0.68 PARP1 (0.62) PARP1KDM4ECA12CA9ALDH1A1
SCHEMBL3423565 0.68 KDM4E (0.50) PARP1GDAKDM4ECA12CA9
SCHEMBL7031558 0.65 PARP1 (0.37) PARP1GDAKDM4ECA12CA9
SCHEMBL29937099 0.65 MAP2 (0.42) PARP1GDAKDM4ECA12CA9
SCHEMBL21230968 0.65 PARP1 (0.37) PARP1GDAKDM4ECA12CA9
SCHEMBL27142990 0.65 MAP2 (0.42) PARP1GDAKDM4ECA12CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1222191-A2 BENZODIAZEPIN DERIVATIVES, THE PRODUCTION AND USE THEREOF BASF AKTIENGESELLSCHAFT (DE) 2002-07-17 EP claimed
WO-2001023386-A2 BENZODIAZEPIN DERIVATIVES, THE PRODUCTION AND USE THEREOF BASF AKTIENGESELLSCHAFT (DE) 2001-04-05 WO claimed
EP-1222191-B1 BENZODIAZEPIN DERIVATIVES, THE PRODUCTION AND USE THEREOF ABBOTT GMBH & CO KG (DE) 2005-11-16 EP disclosed
US-4247296-A Diazo pigments BASF FARBEN & FASERN AG (DE) 1981-01-27 US disclosed