SCHEMBL6201950

SCHEMBL6201950

CCCN(CCC)C(=O)[C@H](C)N

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 4/20 0.44
CA9 Q16790 4/20 0.44
CA2 P00918 3/20 0.44
TSHR P16473 1/20 0.41
MAPK1 P28482 1/20 0.41
ALDH1A1 P00352 1/20 0.39
HPGD P15428 1/20 0.39
TP53 P04637 1/20 0.38
DPP4 P27487 2/20 0.37
CA1 P00915 3/20 0.37
SLC15A1 P46059 1/20 0.34
TDP1 Q9NUW8 2/20 0.34
LMNA P02545 1/20 0.34
HSD17B10 Q99714 1/20 0.34
P2RX1 P51575 2/20 0.33
P2RX4 Q99571 2/20 0.33
P2RX3 P56373 1/20 0.33
BCHE P06276 1/20 0.33
POLB P06746 1/20 0.32
APEX1 P27695 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9873959 1.00 CA12 (0.44) CA12CA9CA2TSHRMAPK1
Trifluoroacetic Acid SCHEMBL9875305 0.87 MLYCD (0.39) CA12CA9CA2TSHRMAPK1
SCHEMBL9875218 0.86 CA12 (0.48) CA12CA9CA2ALDH1A1HPGD
SCHEMBL13944204 0.86 CA12 (0.38) CA12CA9CA2TSHRMAPK1
SCHEMBL22990104 0.82 TSHR (0.37) CA12CA9CA2TSHRMAPK1
SCHEMBL19981940 0.82 DPP4 (0.44) CA12CA9CA2TSHRMAPK1
SCHEMBL4324459 0.81 CA12 (0.32) CA12CA9CA2ALDH1A1DPP4
SCHEMBL9462283 0.80 CA12 (0.48) CA12CA9CA2TSHRMAPK1
SCHEMBL3948078 0.80 DPP4 (0.42) CA12CA9ALDH1A1DPP4CA1
SCHEMBL5438409 0.80 DPP4 (0.42) CA12CA9ALDH1A1DPP4CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1494672-A1 AMINOCARBONYL SUBSTITUTED PYRIDINES, PYRIDAZINES, PYRIMIDINES, PYRAZINES AND TRIAZINES HAVING ANTIANGIOGENIC ACTIVITY Abbott Laboratories (US) 2005-01-12 EP disclosed
WO-2003086398-A1 AMINOCARBONYL SUBSTITUTED PYRIDINES, PYRIDAZINES, PYRIMIDINES, PYRAZINES AND TRIAZINES HAVING ANTIANGIOGENIC ACTIVITY ABBOTT LABORATORIES (US) 2003-10-23 WO disclosed
US-6414013-B1 KINASE INHIBITORS; ANTICANCER AGENTS PHARMACIA & UPJOHN S.P.A. (IT) 2002-07-02 US disclosed