SCHEMBL6202820

SCHEMBL6202820

O=C(CCCNC(=O)c1ccccc1)c1ccc(Br)cc1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.65
NPC1 O15118 3/20 0.57
RAB9A P51151 3/20 0.57
L3MBTL1 Q9Y468 2/20 0.57
NFKB1 P19838 1/20 0.57
CASP3 P42574 1/20 0.57
NFKB2 Q00653 1/20 0.57
RELA Q04206 1/20 0.57
SMN1; SMN2 Q16637 1/20 0.57
SENP8 Q96LD8 1/20 0.57
SENP7 Q9BQF6 1/20 0.57
SENP6 Q9GZR1 1/20 0.57
MEN1 O00255 1/20 0.57
KMT2A Q03164 1/20 0.57
TMEM97 Q5BJF2 1/20 0.56
SIGMAR1 Q99720 1/20 0.56
HDAC4 P56524 4/20 0.56
HDAC1 Q13547 4/20 0.56
HDAC8 Q9BY41 4/20 0.56
HDAC3 O15379 3/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6202779 0.91 NPC1 (0.64) NPC1RAB9AL3MBTL1CASP3SMN1; SMN2
SCHEMBL6223219 0.86 NPC1 (0.58) NPC1RAB9AL3MBTL1HDAC4HDAC1
SCHEMBL2042619 0.84 HDAC1 (0.58) HSP90AA1NPC1RAB9AL3MBTL1MEN1
SCHEMBL6202120 0.81 NPC1 (0.68) NPC1RAB9ANFKB1NFKB2RELA
SCHEMBL6198290 0.80 NPC1 (0.65) NPC1RAB9AL3MBTL1SMN1; SMN2MEN1
SCHEMBL9490115 0.80 HSP90AA1 (0.71) HSP90AA1NPC1RAB9AL3MBTL1NFKB1
SCHEMBL5592824 0.80 PRSS1 (0.68) NPC1RAB9AL3MBTL1SMN1; SMN2MEN1
SCHEMBL9422525 0.80 HSP90AA1 (0.91) HSP90AA1NPC1RAB9ASMN1; SMN2TMEM97
SCHEMBL3030903 0.79 HSP90AA1 (0.69) HSP90AA1NPC1RAB9AL3MBTL1NFKB1
SCHEMBL3034137 0.79 HSP90AA1 (0.65) HSP90AA1NPC1RAB9AL3MBTL1NFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050272036-A1 Ketones ASTRAZENECA AB (SE) 2005-12-08 US disclosed
EP-1549600-A1 KETONES AstraZeneca AB (SE) 2005-07-06 EP disclosed
WO-2004011410-A1 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2004-02-05 WO disclosed