SCHEMBL6203014

SCHEMBL6203014

CC(=O)c1ccccc1F.Fc1ccccc1-c1cocn1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5AP P20292 1/20 0.43
FEN1 P39748 1/20 0.43
ADORA3 P0DMS8 2/20 0.39
ADORA2A P29274 2/20 0.39
NPC1 O15118 6/20 0.39
RAB9A P51151 6/20 0.39
KMT2A Q03164 4/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
ALDH1A1 P00352 3/20 0.39
MEN1 O00255 3/20 0.39
MAPT P10636 2/20 0.39
NFKB1 P19838 1/20 0.39
NFKB2 Q00653 1/20 0.39
RELA Q04206 1/20 0.39
CES2 O00748 1/20 0.39
CES1 P23141 1/20 0.39
KDM4C Q9H3R0 1/20 0.38
SCN9A Q15858 1/20 0.37
RXFP1 Q9HBX9 1/20 0.37
GAA P10253 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6205082 0.83 SCN9A (0.47) ALOX5APFEN1NPC1RAB9AKMT2A
SCHEMBL13461 0.74 CES2 (0.65) FEN1NPC1RAB9AKMT2ASMN1; SMN2
SCHEMBL29593208 0.74 CES2 (0.65) FEN1NPC1RAB9AKMT2ASMN1; SMN2
Hydrochloric Acid SCHEMBL7418290 0.73 CES2 (0.62) FEN1NPC1RAB9AKMT2ASMN1; SMN2
SCHEMBL28925931 0.72 SLC6A3 (0.51) KMT2ASMN1; SMN2ALDH1A1MEN1MAPT
SCHEMBL1515817 0.71 CES2 (0.50) ALOX5APFEN1NPC1RAB9AKMT2A
SCHEMBL29169247 0.69 CES2 (0.58) FEN1NPC1RAB9AKMT2ASMN1; SMN2
Isopropyl Alcohol SCHEMBL29078917 0.68 CES2 (0.56) FEN1NPC1RAB9AKMT2ASMN1; SMN2
Fluorobenzene SCHEMBL28799844 0.68 CES2 (0.56) FEN1NPC1RAB9AKMT2ASMN1; SMN2
SCHEMBL5650569 0.67 SCN9A (0.44) NPC1RAB9AKMT2ASMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501834-A1 TRIARYL-OXY-ARYL-SPIRO-PYRIMIDINE-2, 4, 6-TRIONE METALLOPROTEINASE INHIBITORS Pfizer Products Inc. (US) 2005-02-02 EP disclosed
WO-2003091259-A1 TRIARYL-OXY-ARYL-SPIRO-PYRIMIDINE-2, 4, 6-TRIONE METALLOPROTEINASE INHIBITORS PFIZER PRODUCTS INC. (US) 2003-11-06 WO disclosed