SCHEMBL6203250

SCHEMBL6203250

CCCN(CO)c1nc(Nc2ccccc2)c2[nH]nnc2n1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CCNE2 O96020 2/20 0.38
CCNE1 P24864 2/20 0.38
CDK2 P24941 2/20 0.38
HTR2A P28223 5/20 0.35
HTR2C P28335 5/20 0.35
SRC P12931 1/20 0.35
ADORA3 P0DMS8 2/20 0.33
USP2 O75604 1/20 0.33
ADORA2A P29274 1/20 0.32
NPY5R Q15761 2/20 0.32
MAPK1 P28482 1/20 0.32
PDE4A P27815 1/20 0.31
PDE4B Q07343 1/20 0.31
PDE4C Q08493 1/20 0.31
PDE4D Q08499 1/20 0.31
PDE3B Q13370 1/20 0.31
PDE3A Q14432 1/20 0.31
CRHR1 P34998 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6204147 0.89 CCNE2 (0.40) CCNE2CCNE1CDK2HTR2AHTR2C
SCHEMBL6202094 0.89 HTR2C (0.47) HTR2AHTR2CSRCCRHR1
SCHEMBL6205647 0.88 CDK5 (0.41) CDK2HTR2AHTR2CSRCMAPK1
SCHEMBL6202760 0.85 CDK1 (0.40) CCNE2CCNE1CDK2NPY5RMAPK1
SCHEMBL6203247 0.83 CCNE2 (0.43) CCNE2CCNE1CDK2HTR2AHTR2C
SCHEMBL6205216 0.82 BRAF (0.36) HTR2AHTR2CADORA3
SCHEMBL6204176 0.82 BRAF (0.36) HTR2AHTR2CADORA3
SCHEMBL6203207 0.82 KDM4E (0.36) CCNE2CCNE1CDK2HTR2AHTR2C
SCHEMBL6203171 0.79 CCNE1 (0.37) CCNE2CCNE1CDK2
SCHEMBL6204529 0.79 CCNE2 (0.44) CCNE2CCNE1CDK2HTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1539760-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2005-06-15 EP disclosed
WO-2004018473-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2004-03-04 WO disclosed