SCHEMBL6202760

SCHEMBL6202760

CCCN(CO)c1nc(NCc2ccccc2)c2[nH]nnc2n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 3/20 0.40
CDK5 Q00535 1/20 0.40
PDE4A P27815 2/20 0.38
PDE4B Q07343 2/20 0.38
PDE4C Q08493 2/20 0.38
PDE4D Q08499 2/20 0.38
CDK2 P24941 4/20 0.38
CCNE2 O96020 3/20 0.38
CCNE1 P24864 3/20 0.38
PPARG P37231 1/20 0.37
PRUNE1 Q86TP1 1/20 0.36
APP P05067 2/20 0.36
BCHE P06276 2/20 0.36
ACHE P22303 2/20 0.36
LMNA P02545 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
TSHR P16473 1/20 0.36
MAPK1 P28482 1/20 0.36
AGTR1 P30556 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6203171 0.86 CCNE1 (0.37) CDK5CDK2CCNE2CCNE1AGTR1
SCHEMBL6203250 0.85 CCNE2 (0.38) PDE4APDE4BPDE4CPDE4DCDK2
SCHEMBL6202754 0.84 CDK5 (0.43) CDK1CDK5PDE4APDE4BPDE4C
SCHEMBL6205608 0.84 PARP1 (0.36) PDE4APDE4BPDE4CPDE4DPRUNE1
SCHEMBL7013199 0.82 CDK1 (0.39) CDK1CDK5PDE4APDE4BPDE4C
SCHEMBL6201142 0.80 CDK1 (0.46) CDK1CDK5PDE4APDE4BPDE4C
SCHEMBL6204811 0.79 PRUNE1 (0.32) PDE4DCDK2CCNE1PRUNE1TSHR
SCHEMBL6204719 0.78 PGK1 (0.33)
SCHEMBL6203495 0.78 PRUNE1 (0.35) CDK1CDK5PDE4DCDK2CCNE2
SCHEMBL6205414 0.77 HMGCR (0.32) PRUNE1EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1539760-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2005-06-15 EP claimed
WO-2004018473-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2004-03-04 WO claimed
EP-1539760-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2005-06-15 EP disclosed
WO-2004018473-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2004-03-04 WO disclosed