SCHEMBL6203315

SCHEMBL6203315

CC=C(CS(=O)(=O)c1ccccc1Br)OC(=O)c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLCG1 P19174 1/20 0.44
POLB P06746 3/20 0.38
TSHR P16473 2/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA4 P22748 1/20 0.36
CA6 P23280 1/20 0.36
HSD11B1 P28845 2/20 0.35
ALDH1A1 P00352 2/20 0.35
LMNA P02545 2/20 0.35
HSD17B10 Q99714 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
KDM4E B2RXH2 1/20 0.34
F2 P00734 1/20 0.34
CES2 O00748 1/20 0.34
CES1 P23141 1/20 0.34
RECQL P46063 2/20 0.34
NPC1 O15118 1/20 0.34
HPGD P15428 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28911450 0.75 PLCG1 (0.56) PLCG1POLBCA1CA2CA4
SCHEMBL27933271 0.75 PLCG1 (0.51) PLCG1POLBTSHRCA1CA2
SCHEMBL5799667 0.74 TSHR (0.52) TSHRCA1CA2ALDH1A1LMNA
SCHEMBL5799668 0.74 TSHR (0.52) TSHRCA1CA2ALDH1A1LMNA
SCHEMBL9183020 0.72 TDP1 (0.48) POLBTSHRCA1CA2ALDH1A1
SCHEMBL15917034 0.69 HSD11B1 (0.62) PLCG1POLBCA1CA2CA4
SCHEMBL6203312 0.69 PLCG1 (0.45) PLCG1POLBTSHRCA1CA2
SCHEMBL11226379 0.69 PLCG1 (0.60) PLCG1POLBCA1CA2CA4
SCHEMBL27933035 0.67 HSD11B1 (0.63) PLCG1CA1CA2CA4CA6
SCHEMBL27638996 0.67 PLCG1 (0.62) PLCG1POLBCA1CA2CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1425279-A4 METHOD FOR THE PREPARATION OF CRYSTALLINE TETRAHYDROBENZOTHIEPINES SEARLE LLC (US) 2005-10-26 EP disclosed
EP-1425279-A2 METHOD FOR THE PREPARATION OF CRYSTALLINE TETRAHYDROBENZOTHIEPINES G.D. Searle LLC (US) 2004-06-09 EP disclosed
WO-2003022804-A9 METHOD FOR THE PREPARATION OF CRYSTALLINE TETRAHYDROBENZOTHIEPINES SEARLE LLC (US) 2003-12-18 WO disclosed
WO-2003022804-A2 METHOD FOR THE PREPARATION OF CRYSTALLINE TETRAHYDROBENZOTHIEPINES G.D. SEARLE LLC (US) 2003-03-20 WO disclosed