SCHEMBL6203322

SCHEMBL6203322

COC(OC)c1cccc(Cl)c1

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 1/20 0.53
SLC6A2 P23975 1/20 0.42
SLC6A4 P31645 1/20 0.42
SLC6A3 Q01959 1/20 0.42
ACP3 P15309 1/20 0.42
PDE1B Q01064 1/20 0.40
HSD17B2 P37059 1/20 0.40
OPRM1 P35372 2/20 0.39
OPRD1 P41143 2/20 0.39
OPRK1 P41145 2/20 0.39
OPRL1 P41146 2/20 0.39
PNMT P11086 1/20 0.38
ALDH1A1 P00352 1/20 0.38
TSHR P16473 1/20 0.38
RELA Q04206 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17864868 0.84 HDAC4 (0.38) AOC3
SCHEMBL3096347 0.81 AOC3 (0.56) AOC3SLC6A2SLC6A4SLC6A3ACP3
SCHEMBL11395224 0.81 AOC3 (0.51) AOC3SLC6A2SLC6A4SLC6A3ACP3
SCHEMBL6204741 0.79 AOC3 (0.50) AOC3SLC6A2SLC6A4SLC6A3ACP3
SCHEMBL16953022 0.79 AOC3 (0.50) AOC3SLC6A2SLC6A4SLC6A3ACP3
SCHEMBL10861290 0.79 AOC3 (0.42) AOC3SLC6A2SLC6A4SLC6A3ACP3
SCHEMBL6204740 0.79 AOC3 (0.50) AOC3SLC6A2SLC6A4SLC6A3ACP3
SCHEMBL6155751 0.78 AOC3 (0.45) AOC3SLC6A2SLC6A4SLC6A3ACP3
SCHEMBL11403406 0.77 TSHR (0.42) AOC3SLC6A4TSHR
SCHEMBL24615882 0.76 AOC3 (0.64) AOC3SLC6A2SLC6A4SLC6A3ACP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104230879-B A kind of 2-((4R, 6S)-6-formoxyl-2,2-disubstituted-1,3-dioxane-4-base) acetas preparation method 新发药业有限公司 2016-08-24 CN disclosed
CN-105722823-A NOVEL CYTOCHROME P450 INHIBITORS AND THEIR METHOD OF USE 科尔泰多公众股份公司 2016-06-29 CN disclosed
CN-104230879-A Simple and convenient preparation method of 2-((4R,6S)-6-formyl-2,2-disubstituted-1,3-dioxane-4-yl)acetate XINFA PHARMACEUTICAL CO LTD 2014-12-24 CN disclosed
EP-1506175-A1 N-SUBSTITUTED TRICYCLIC 3-AMINOPYRAZOLES AS PDGF RECEPTOR INHIBITORS JANSSEN PHARMACEUTICA N.V. (BE) 2005-02-16 EP disclosed
WO-2003097609-A1 N-SUBSTITUTED TRICYCLIC 3-AMINOPYRAZOLES AS PDFG RECEPTOR INHIBITORS JANSSEN PHARMACEUTICA N.V. (BE) 2003-11-27 WO disclosed
EP-0918757-A1 8-HYDROCARBYL SUBSTITUTED BENZODIZOCINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS PROTEIN KINASE C (=PKC) MODULATORS GEORGETOWN UNIVERSITY (US) 1999-06-02 EP disclosed
WO-1997043268-A1 8-HYDROCARBYL SUBSTITUTED BENZODIZOCINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS PROTEIN KINASE C (=PKC) MODULATORS GEORGETOWN UNIVERSITY (US) 1997-11-20 WO disclosed
US-4629737-A HYPOGLYCEMIC AGENTS; DIETETICS BEECHAM GROUP P.L.C. (GB) 1986-12-16 US disclosed
EP-0099707-B1 2-AMINOETHYL ETHER DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM BEECHAM GROUP PLC (GB) 1986-12-10 EP disclosed
EP-0099707-A1 2-Aminoethyl ether derivatives, processes for their preparation and pharmaceutical compositions containing them BEECHAM GROUP PLC (GB) 1984-02-01 EP disclosed
US-4246021-A Imidazole derivatives MAY & BAKER LIMITED (GB) 1981-01-20 US disclosed