SCHEMBL6203420

SCHEMBL6203420

CC(=O)c1ccccc1CNc1nc(N(CCO)C(C)C)nc2c1N(C(C)C)NN2C(C)C

nearest known ligand 0.33

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 2/20 0.33
CDK5 Q00535 1/20 0.33
CDK2 P24941 6/20 0.33
CCNE2 O96020 5/20 0.33
CCNE1 P24864 5/20 0.33
HCRTR1 O43613 1/20 0.31
HCRTR2 O43614 1/20 0.31
PDE5A O76074 1/20 0.30
PDE6C P51160 1/20 0.30
PDE4D Q08499 1/20 0.30
CCNB2 O95067 1/20 0.30
CCNB1 P14635 1/20 0.30
CCNB3 Q8WWL7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6201113 0.84 CDK1 (0.46) CDK1CDK5CDK2CCNE2CCNE1
SCHEMBL6205622 0.82 CCNE2 (0.35) CDK1CDK5CDK2CCNE2CCNE1
SCHEMBL6202735 0.81 CCNE1 (0.44) CDK2CCNE2CCNE1
SCHEMBL6203391 0.80 CCNE2 (0.31) CDK1CDK5CDK2CCNE2CCNE1
SCHEMBL3444131 0.80 CDK1 (0.46) CDK1CDK5CDK2CCNE2CCNE1
SCHEMBL6205419 0.78 CCNE1 (0.36) CDK1CDK5CDK2CCNE2CCNE1
SCHEMBL3444674 0.78 CDK2 (0.42) CDK1CDK5CDK2CCNE2CCNE1
SCHEMBL3445521 0.78 CDK2 (0.37) CDK1CDK5CDK2CCNE2CCNE1
SCHEMBL3444730 0.77 CDK2 (0.47) CDK1CDK5CDK2CCNE2CCNE1
SCHEMBL6202208 0.77 CDK1 (0.33) CDK1CDK5CDK2CCNE2CCNE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1539760-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2005-06-15 EP disclosed
WO-2004018473-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2004-03-04 WO disclosed