SCHEMBL6202208

SCHEMBL6202208

CC(=O)c1ccccc1CNc1nc(N(CCO)C(C)C)nc2nn[nH]c12

nearest known ligand 0.33

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 1/20 0.33
CDK5 Q00535 1/20 0.33
CCNE2 O96020 1/20 0.32
CCNE1 P24864 1/20 0.32
CDK2 P24941 1/20 0.32
JAK2 O60674 2/20 0.31
JAK1 P23458 2/20 0.31
TYK2 P29597 2/20 0.31
JAK3 P52333 2/20 0.31
PDE5A O76074 1/20 0.31
PDE6C P51160 1/20 0.31
PDE4D Q08499 1/20 0.31
HCRTR1 O43613 1/20 0.30
HCRTR2 O43614 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6204605 0.87 TSHR (0.32) CDK1CDK5CCNE2CCNE1CDK2
SCHEMBL6203326 0.86 CDK2 (0.38) CDK1CDK5CCNE2CCNE1CDK2
SCHEMBL6201142 0.84 CDK1 (0.46) CDK1CDK5CCNE2CCNE1CDK2
SCHEMBL6203806 0.82 STAT3 (0.36) CDK1CDK5CCNE2CCNE1CDK2
SCHEMBL6205328 0.82 PARP1 (0.36) CDK1CDK5CCNE2CCNE1CDK2
SCHEMBL6204274 0.79 CCR4 (0.33) CCNE2CCNE1CDK2
SCHEMBL6204529 0.78 CCNE2 (0.44) CDK1CDK5CCNE2CCNE1CDK2
SCHEMBL6203855 0.78 CCNE1 (0.34) CDK1CDK5CCNE2CCNE1CDK2
SCHEMBL3444027 0.77 CDK2 (0.45) CDK1CDK5CCNE1CDK2JAK1
SCHEMBL3444871 0.77 CDK1 (0.45) CDK1CDK5CCNE2CCNE1CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1539760-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2005-06-15 EP claimed
WO-2004018473-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2004-03-04 WO claimed
EP-1539760-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2005-06-15 EP disclosed
WO-2004018473-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2004-03-04 WO disclosed