SCHEMBL6204433

SCHEMBL6204433

COc1ccc(CC(=O)c2cccc(Br)c2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.54
LMNA P02545 2/20 0.54
NPC1 O15118 2/20 0.54
HTT P42858 2/20 0.54
HPGD P15428 2/20 0.53
USP2 O75604 1/20 0.51
TP53 P04637 1/20 0.51
HSP90AA1 P07900 1/20 0.50
SLC2A1 P11166 1/20 0.49
ALDH1A1 P00352 2/20 0.49
TDP1 Q9NUW8 1/20 0.49
KMT2A Q03164 3/20 0.49
MEN1 O00255 2/20 0.49
CYP3A4 P08684 2/20 0.49
RAB9A P51151 1/20 0.49
ATM Q13315 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
CYP1A2 P05177 1/20 0.48
CYP2D6 P10635 1/20 0.48
CYP2C19 P33261 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27572327 0.86 ALDH1A1 (0.63) MAPTLMNANPC1HTTHPGD
SCHEMBL27626615 0.84 PARP1 (0.52) MAPTLMNANPC1TP53ALDH1A1
SCHEMBL16162272 0.84 NPC1 (0.55) MAPTLMNANPC1HTTHPGD
SCHEMBL28438923 0.84 RAB9A (0.61) MAPTLMNANPC1HTTHPGD
SCHEMBL12916784 0.82 NPC1 (0.63) MAPTNPC1HTTSLC2A1ALDH1A1
SCHEMBL7854504 0.81 KMT2A (0.64) MAPTLMNANPC1HTTUSP2
SCHEMBL6203838 0.81 KMT2A (0.64) MAPTLMNANPC1HTTUSP2
SCHEMBL931177 0.81 MAPT (0.57) MAPTNPC1ALDH1A1KMT2AMEN1
SCHEMBL571063 0.81 USP2 (0.69) MAPTLMNANPC1HTTUSP2
SCHEMBL22773277 0.80 ALDH1A1 (0.60) MAPTLMNANPC1TP53ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050272036-A1 Ketones ASTRAZENECA AB (SE) 2005-12-08 US disclosed
CN-1681763-A Chemical compounds ASTRAZENECA AB (SE) 2005-10-12 CN disclosed
EP-1549600-A1 KETONES AstraZeneca AB (SE) 2005-07-06 EP disclosed
WO-2004011410-A1 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2004-02-05 WO disclosed