SCHEMBL6204828

SCHEMBL6204828

O[C@H](CNc1nc(Cl)nc2nn[nH]c12)c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.40
HPGD P15428 1/20 0.39
MAPK1 P28482 1/20 0.39
KDM4E B2RXH2 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
NPC1 O15118 1/20 0.39
FAAH O00519 3/20 0.37
AOC3 Q16853 3/20 0.37
AURKA O14965 1/20 0.35
RPS6KB1 P23443 1/20 0.35
HTT P42858 1/20 0.35
ROCK2 O75116 1/20 0.35
ROCK1 Q13464 1/20 0.35
ADRB2 P07550 1/20 0.34
CDK1 P06493 1/20 0.34
CDK5 Q00535 1/20 0.34
BCAT2 O15382 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7711077 0.81 SMN1; SMN2 (0.53) CYP2D6CDK1
SCHEMBL3444344 0.78 PDE5A (0.54) CYP2D6HPGDMAPK1CDK1
SCHEMBL3445624 0.78 EGFR (0.39) HPGDAURKARPS6KB1
SCHEMBL3445625 0.78 EGFR (0.39) HPGDAURKARPS6KB1
SCHEMBL17799994 0.74 APP (0.58) CYP2D6HPGDMAPK1KDM4EL3MBTL1
SCHEMBL7334685 0.70 HPGD (0.46) CYP2D6HPGDMAPK1KDM4EL3MBTL1
SCHEMBL654721 0.69 L3MBTL1 (0.49) CYP2D6HPGDMAPK1KDM4EL3MBTL1
SCHEMBL22401301 0.68 KDM4E (0.47) CYP2D6HPGDMAPK1KDM4EL3MBTL1
SCHEMBL7711075 0.68 CDK1 (0.69) MAPK1KDM4ENPC1CDK1CDK5
SCHEMBL6298554 0.67 CYP2D6 (0.54) CYP2D6HPGDMAPK1KDM4EL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1539760-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2005-06-15 EP claimed
WO-2004018473-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2004-03-04 WO claimed
EP-1539760-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2005-06-15 EP disclosed
WO-2004018473-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2004-03-04 WO disclosed