SCHEMBL6204848

SCHEMBL6204848

CC(C)N(CCO)c1nc(Nc2ccc(Cl)c(C(=O)O)c2)c2[nH]nnc2n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK5 Q00535 3/20 0.40
CDK5R1 Q15078 3/20 0.40
CDK1 P06493 2/20 0.40
MAPT P10636 5/20 0.34
TDP1 Q9NUW8 4/20 0.34
KDM4E B2RXH2 3/20 0.34
POLB P06746 3/20 0.34
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
ALDH1A1 P00352 2/20 0.34
CCNA2 P20248 2/20 0.34
CDK2 P24941 2/20 0.34
CCNA1 P78396 2/20 0.34
CCNB2 O95067 1/20 0.34
CCNE2 O96020 1/20 0.34
NTRK1 P04629 1/20 0.34
INSR P06213 1/20 0.34
CCNB1 P14635 1/20 0.34
PRKACA P17612 1/20 0.34
PRKACG P22612 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6205471 0.93 CDK5 (0.40) CDK5CDK5R1CDK1KDM4EALDH1A1
SCHEMBL6201043 0.90 CDK1 (0.40) CDK5CDK5R1CDK1MAPTALDH1A1
SCHEMBL6204246 0.86 BRAF (0.35) CDK5CDK5R1CDK2CCNE2CCNE1
SCHEMBL6204587 0.85 BRAF (0.35) CDK5CDK5R1CDK2CCNE2CCNE1
SCHEMBL6205187 0.84 HTR2C (0.42) CDK5CDK5R1CDK1CDK2CCNE2
SCHEMBL6202531 0.83 CDK5 (0.46) CDK5CDK5R1CDK1MAPTTDP1
SCHEMBL6204529 0.82 CCNE2 (0.44) CDK5CDK5R1CDK1CDK2CCNE2
SCHEMBL6203534 0.80 CCNE2 (0.46) CDK1CDK2CCNE2CCNE1
SCHEMBL6204534 0.79 CLK1 (0.36) CDK5CDK5R1CDK1MAPTTDP1
SCHEMBL3445187 0.78 CDK1 (0.61) CDK5CDK5R1CDK1MAPTTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1539760-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2005-06-15 EP claimed
WO-2004018473-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2004-03-04 WO claimed