SCHEMBL6204587

SCHEMBL6204587

CC(C)N(CCO)c1nc(Nc2ccc(N)c(Cl)c2)c2[nH]nnc2n1

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
BRAF P15056 2/20 0.35
CDK5 Q00535 2/20 0.33
CDK5R1 Q15078 2/20 0.33
ATM Q13315 1/20 0.33
CCNE2 O96020 2/20 0.31
CCNE1 P24864 2/20 0.31
CDK2 P24941 2/20 0.31
HTR2A P28223 1/20 0.31
HTR2C P28335 1/20 0.31
ERBB2 P04626 2/20 0.30
KCNH2 Q12809 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6204246 0.93 BRAF (0.35) BRAFCDK5CDK5R1ATMCCNE2
SCHEMBL6205471 0.86 CDK5 (0.40) BRAFCDK5CDK5R1ATMCCNE2
SCHEMBL6205187 0.86 HTR2C (0.42) CDK5CDK5R1ATMCCNE2CCNE1
SCHEMBL6202531 0.85 CDK5 (0.46) BRAFCDK5CDK5R1ATMCCNE2
SCHEMBL6204534 0.85 CLK1 (0.36) BRAFCDK5CDK5R1ATM
SCHEMBL6204848 0.85 CDK5 (0.40) CDK5CDK5R1ATMCCNE2CCNE1
SCHEMBL6203534 0.82 CCNE2 (0.46) CCNE2CCNE1CDK2HTR2AHTR2C
SCHEMBL6204529 0.82 CCNE2 (0.44) CDK5CDK5R1ATMCCNE2CCNE1
SCHEMBL6205216 0.82 BRAF (0.36) BRAFHTR2AHTR2C
SCHEMBL6204524 0.80 CCNE2 (0.34) CDK5CDK5R1CCNE2CCNE1CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1539760-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2005-06-15 EP claimed
WO-2004018473-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2004-03-04 WO claimed
EP-1539760-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2005-06-15 EP disclosed
WO-2004018473-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2004-03-04 WO disclosed