SCHEMBL6204534

SCHEMBL6204534

CC(C)N(CCO)c1nc(Nc2cc(N)cc(Cl)c2)c2[nH]nnc2n1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CLK1 P49759 10/20 0.36
CDK1 P06493 2/20 0.36
CCNB1 P14635 2/20 0.36
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 1/20 0.36
CCNB2 O95067 1/20 0.36
ALDH1A1 P00352 1/20 0.36
TP53 P04637 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
MAPT P10636 1/20 0.36
CYP2C9 P11712 1/20 0.36
HPGD P15428 1/20 0.36
TSHR P16473 1/20 0.36
MAPK1 P28482 1/20 0.36
KMT2A Q03164 1/20 0.36
CCNB3 Q8WWL7 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
CDK5 Q00535 1/20 0.33
ATM Q13315 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6202531 0.86 CDK5 (0.46) CDK1CCNB1KDM4EMEN1CCNB2
SCHEMBL6205187 0.86 HTR2C (0.42) CDK1CDK5ATMCDK5R1
SCHEMBL6204246 0.85 BRAF (0.35) CDK5ATMCDK5R1BRAF
SCHEMBL6204587 0.85 BRAF (0.35) CDK5ATMCDK5R1BRAF
SCHEMBL6204529 0.82 CCNE2 (0.44) CDK1CDK5ATMCDK5R1
SCHEMBL6203534 0.80 CCNE2 (0.46) CDK1MAPK1
SCHEMBL6205469 0.80
SCHEMBL6205471 0.79 CDK5 (0.40) CDK1CCNB1KDM4ECCNB2ALDH1A1
SCHEMBL6204848 0.79 CDK5 (0.40) CDK1CCNB1KDM4EMEN1CCNB2
SCHEMBL6204524 0.76 CCNE2 (0.34) CDK1CCNB1CDK5CDK5R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1539760-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2005-06-15 EP claimed
WO-2004018473-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2004-03-04 WO claimed
EP-1539760-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2005-06-15 EP disclosed
WO-2004018473-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2004-03-04 WO disclosed