SCHEMBL6204877

SCHEMBL6204877

CCCCCN(CCc1ccc(Oc2ccc(C(N)=O)cn2)c(C)c1)c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 15/20 0.43
OPRK1 P41145 12/20 0.43
OPRD1 P41143 11/20 0.43
GRIN2D O15399 1/20 0.42
GRIN3B O60391 1/20 0.42
SLC6A2 P23975 1/20 0.42
SLC6A3 Q01959 1/20 0.42
GRIN1 Q05586 1/20 0.42
KCNH2 Q12809 1/20 0.42
GRIN2A Q12879 1/20 0.42
GRIN2B Q13224 1/20 0.42
ROCK1 Q13464 1/20 0.42
GRIN2C Q14957 1/20 0.42
GRIN3A Q8TCU5 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6203886 0.90 OPRM1 (0.38) OPRM1OPRK1OPRD1GRIN2DGRIN3B
SCHEMBL6203883 0.88 OPRM1 (0.43) OPRM1OPRK1OPRD1GRIN2DGRIN3B
SCHEMBL6224838 0.83 OPRM1 (0.42) OPRM1OPRK1OPRD1GRIN2DGRIN3B
SCHEMBL6227482 0.82 NR1H3 (0.43) OPRM1OPRK1OPRD1GRIN2DGRIN3B
SCHEMBL6228196 0.82 OPRM1 (0.42) OPRM1OPRK1OPRD1GRIN2DGRIN3B
SCHEMBL6224928 0.82 OPRM1 (0.38) OPRM1OPRK1OPRD1GRIN2DGRIN3B
SCHEMBL3700138 0.80 OPRM1 (0.56) OPRM1OPRK1OPRD1GRIN2DGRIN3B
SCHEMBL6224920 0.80 OPRM1 (0.43) OPRM1OPRK1OPRD1GRIN2DGRIN3B
SCHEMBL3690747 0.79 OPRM1 (0.52) OPRM1OPRK1OPRD1GRIN2DGRIN3B
SCHEMBL3695129 0.78 NNMT (0.48) OPRM1OPRK1OPRD1GRIN2DGRIN3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1562595-A1 DIARYL ETHERS AS OPIOID RECEPTOR ANTAGONISTS ELI LILLY AND COMPANY (US) 2005-08-17 EP disclosed
WO-2004026305-A1 DIARYL ETHERS AS OPIOID RECEPTOR ANTAGONIST ELI LILLY AND COMPANY (US) 2004-04-01 WO disclosed