SCHEMBL6205037

SCHEMBL6205037

CC(=O)Oc1ccc(C(=O)n2c(C)c(CC(=O)O)c3ccccc32)cc1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 3/20 0.71
PTGS2 P35354 3/20 0.71
PTGS1 P23219 2/20 0.71
LMNA P02545 2/20 0.64
CYP1A2 P05177 2/20 0.64
CYP2D6 P10635 2/20 0.64
CYP2C9 P11712 2/20 0.64
HIF1A Q16665 2/20 0.64
NPSR1 Q6W5P4 2/20 0.64
TSHR P16473 1/20 0.64
NFKB1 P19838 1/20 0.64
AKR1C3 P42330 6/20 0.61
AKR1C2 P52895 6/20 0.61
AKR1C4 P17516 2/20 0.57
AKR1C1 Q04828 2/20 0.57
KDM4E B2RXH2 1/20 0.57
MEN1 O00255 1/20 0.57
PTGES O14684 1/20 0.57
ABCC3 O15438 1/20 0.57
ABCC4 O15439 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13802380 0.88 AKR1C3 (0.78) ABCB1PTGS2PTGS1LMNACYP1A2
Delmetacin SCHEMBL286727 0.86 ABCB1 (0.82) ABCB1PTGS2PTGS1LMNACYP1A2
SCHEMBL5646081 0.86 PTGS2 (0.54) ABCB1PTGS2PTGS1LMNACYP1A2
SCHEMBL13802409 0.85 ABCB1 (0.81) ABCB1PTGS2PTGS1LMNACYP1A2
SCHEMBL4205369 0.85 ABCB1 (0.69) ABCB1PTGS2PTGS1LMNACYP1A2
SCHEMBL4213009 0.84 ABCB1 (0.68) ABCB1PTGS2PTGS1LMNACYP1A2
SCHEMBL6206650 0.84 ABCB1 (0.79) ABCB1PTGS2PTGS1LMNACYP1A2
SCHEMBL2237296 0.83 ABCB1 (1.00) ABCB1PTGS2PTGS1LMNACYP1A2
SCHEMBL6206463 0.83 ABCB1 (0.77) ABCB1PTGS2PTGS1LMNACYP1A2
SCHEMBL4209260 0.80 LMNA (0.71) ABCB1PTGS2PTGS1LMNACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1600440-A1 INDOLE DERIVATIVE COMPOUNDS AND DRUGS CONTAINING THE COMPOUNDS AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO., LTD. (JP) 2005-11-30 EP disclosed