SCHEMBL6205310

SCHEMBL6205310

O=C(Nc1ccc(S(=O)(=O)N(Cc2ccccc2)C2CCNCC2)c2ccccc12)c1ccccc1

nearest known ligand 0.61

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CCR8 P51685 16/20 0.61
SMYD3 Q9H7B4 1/20 0.41
HDAC8 Q9BY41 2/20 0.41
HDAC6 Q9UBN7 2/20 0.41
SLC6A2 P23975 1/20 0.41
SLC6A4 P31645 1/20 0.41
SLC6A3 Q01959 1/20 0.41
KCNH2 Q12809 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6203974 0.81 SLC6A2 (0.42) CCR8SMYD3HDAC8HDAC6SLC6A2
SCHEMBL1338876 0.80 CCR8 (0.60) CCR8
SCHEMBL6409599 0.77 SMYD3 (0.39) CCR8SMYD3HDAC8HDAC6SLC6A2
SCHEMBL6248251 0.76 CCR8 (0.57) CCR8
SCHEMBL1338154 0.76 CCR8 (1.00) CCR8
SCHEMBL6438547 0.75 CCR8 (0.55) CCR8
SCHEMBL6204924 0.75 CCR8 (0.55) CCR8
SCHEMBL6365514 0.75 CCR8 (0.54) CCR8
SCHEMBL6408725 0.74 CCR8 (0.54) CCR8
SCHEMBL6364712 0.74 CCR8 (0.54) CCR8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1590327-A1 CCR8 INHIBITORS MILLENNIUM PHARMACEUTICALS, INC. (US) 2005-11-02 EP disclosed
EP-1581511-A1 CCR8 INHIBITORS MILLENNIUM PHARMACEUTICALS, INC. (US) 2005-10-05 EP disclosed
WO-2004058709-A1 CCR8 INHIBITORS MILLENNIUM PHARMACEUTICALS, INC. (US) 2004-07-15 WO disclosed
WO-2004058736-A1 CCR8 INHIBITORS MILLENNIUM PHARMACEUTICALS, INC. (US) 2004-07-15 WO disclosed