SCHEMBL6409599

SCHEMBL6409599

COCNC(=O)c1ccc(S(=O)(=O)N(Cc2ccccc2)C2CCNCC2)c2ccccc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
SLC6A2 P23975 3/20 0.38
SLC6A4 P31645 3/20 0.38
SLC6A3 Q01959 1/20 0.38
KCNH2 Q12809 1/20 0.38
DCUN1D1 Q96GG9 1/20 0.36
CCR8 P51685 1/20 0.36
HTR2A P28223 2/20 0.35
KMT2A Q03164 2/20 0.35
MAPK1 P28482 2/20 0.35
KDM4E B2RXH2 1/20 0.35
HTT P42858 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
HSD17B10 Q99714 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
NMT1 P30419 1/20 0.35
MMP1 P03956 2/20 0.35
MMP9 P14780 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6203974 0.84 SLC6A2 (0.42) SMYD3L3MBTL1SLC6A2SLC6A4SLC6A3
SCHEMBL6205310 0.77 CCR8 (0.61) SMYD3SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL1339959 0.70 KMT2A (0.53) CCR8KMT2AHTTSMN1; SMN2MEN1
SCHEMBL6416674 0.69 CYP1A2 (0.43) SLC6A2SLC6A4SLC6A3KCNH2CCR8
SCHEMBL2958329 0.67 CNR2 (0.57) SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL6205468 0.67 SLC6A4 (0.42) SLC6A2SLC6A4SLC6A3KCNH2CCR8
SCHEMBL6365514 0.67 CCR8 (0.54) CCR8
SCHEMBL24392681 0.66 SLC6A2 (0.53) SMYD3SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL6204924 0.66 CCR8 (0.55) CCR8
SCHEMBL6254437 0.66 CCR8 (0.57) CCR8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1581511-A1 CCR8 INHIBITORS MILLENNIUM PHARMACEUTICALS, INC. (US) 2005-10-05 EP disclosed
WO-2004058736-A1 CCR8 INHIBITORS MILLENNIUM PHARMACEUTICALS, INC. (US) 2004-07-15 WO disclosed