SCHEMBL620590

SCHEMBL620590

CC(C)(C)[S@@+]([O-])/N=C/Cc1ccccc1F

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GPR3 P46089 1/20 0.38
TAAR1 Q96RJ0 3/20 0.35
RIPK1 Q13546 2/20 0.34
IDO1 P14902 2/20 0.33
AOC3 Q16853 1/20 0.33
MAOA P21397 1/20 0.31
MAOB P27338 1/20 0.31
LMNA P02545 2/20 0.31
ALDH1A1 P00352 2/20 0.31
USP2 O75604 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17028760 1.00 GPR3 (0.38) GPR3TAAR1RIPK1IDO1AOC3
SCHEMBL17028761 1.00 GPR3 (0.38) GPR3TAAR1RIPK1IDO1AOC3
SCHEMBL15994994 0.89 RIPK1 (0.35) GPR3RIPK1
SCHEMBL17749309 0.89 RIPK1 (0.35) GPR3RIPK1
SCHEMBL15994995 0.89 RIPK1 (0.35) GPR3RIPK1
SCHEMBL17028752 0.87 NPC1 (0.38) RIPK1MAOBLMNAALDH1A1
SCHEMBL30681392 0.87 GPR3 (0.30) GPR3
SCHEMBL2582230 0.86 TAAR1 (0.40) GPR3TAAR1RIPK1IDO1AOC3
SCHEMBL15820811 0.81 IDO1 (0.37) RIPK1IDO1MAOB
SCHEMBL15820812 0.81 IDO1 (0.37) RIPK1IDO1MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3353163-A1 2,3,4,5-TETRAHYDROPYRIDIN-6-AMINE DERIVATIVES Janssen Pharmaceutica, N.V. (BE) 2018-08-01 EP disclosed
EP-3271355-A1 BACE1 INHIBITORS F. Hoffmann-La Roche AG (CH) 2018-01-24 EP disclosed
WO-2017050978-A1 2,3,4,5-TETRAHYDROPYRIDIN-6-AMINE DERIVATIVES JANSSEN PHARMACEUTICA NV (BE) 2017-03-30 WO disclosed
WO-2016150785-A1 BACE1 INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2016-09-29 WO disclosed
WO-2011138293-A1 2,5,6,7-TETRAHYDRO-[1,4]OXAZEPIN-3-YLAMINE OR 2,3,6,7-TETRAHYDRO-[1,4]OXAZEPIN-5-YLAMINE COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2011-11-10 WO disclosed