SCHEMBL6206329

SCHEMBL6206329

CCCC(=O)N(C1CCNCC1C)S(=O)(=O)c1ccc(C(N)=O)c2ccccc12

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 12/20 0.37
SLC6A4 P31645 12/20 0.37
SLC6A3 Q01959 7/20 0.37
KCNH2 Q12809 3/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
CNR1 P21554 1/20 0.32
CCR8 P51685 1/20 0.32
CYP2D6 P10635 2/20 0.32
CHEK1 O14757 1/20 0.32
RPS6KB1 P23443 1/20 0.31
HTR6 P50406 1/20 0.31
PARP1 P09874 1/20 0.31
PARP2 Q9UGN5 1/20 0.31
ACVR1 Q04771 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6204001 0.85 SLC6A4 (0.39) SLC6A2SLC6A4SLC6A3KCNH2ALDH1A1
SCHEMBL6361502 0.81 CCR8 (0.55) CCR8
SCHEMBL6206397 0.81 CCR8 (0.55) CCR8
SCHEMBL6437668 0.81 CCR8 (0.55) CCR8
SCHEMBL4951730 0.78 CCR8 (0.53) CCR8
SCHEMBL4951725 0.78 CCR8 (0.53) CCR8
SCHEMBL6205468 0.76 SLC6A4 (0.42) SLC6A2SLC6A4SLC6A3KCNH2CCR8
SCHEMBL6416674 0.72 CYP1A2 (0.43) SLC6A2SLC6A4SLC6A3KCNH2LMNA
SCHEMBL6204231 0.70 CCR8 (0.51) ALDH1A1LMNACCR8
SCHEMBL6204695 0.70 SLC6A2 (0.40) SLC6A2SLC6A4SLC6A3KCNH2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1590327-A1 CCR8 INHIBITORS MILLENNIUM PHARMACEUTICALS, INC. (US) 2005-11-02 EP disclosed
EP-1581511-A1 CCR8 INHIBITORS MILLENNIUM PHARMACEUTICALS, INC. (US) 2005-10-05 EP disclosed
WO-2004058709-A1 CCR8 INHIBITORS MILLENNIUM PHARMACEUTICALS, INC. (US) 2004-07-15 WO disclosed
WO-2004058736-A1 CCR8 INHIBITORS MILLENNIUM PHARMACEUTICALS, INC. (US) 2004-07-15 WO disclosed