SCHEMBL6416674

SCHEMBL6416674

CCCC(=O)N(C1CCNCC1)S(=O)(=O)c1ccc(C(=O)Nc2ccccc2)c2ccccc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
MAPT P10636 1/20 0.43
CYP2C9 P11712 1/20 0.43
HPGD P15428 1/20 0.43
CYP2C19 P33261 1/20 0.43
ATM Q13315 1/20 0.43
CCR8 P51685 9/20 0.40
KMT2A Q03164 3/20 0.39
HTT P42858 2/20 0.39
SLC6A2 P23975 3/20 0.39
SLC6A4 P31645 3/20 0.39
SLC6A3 Q01959 3/20 0.39
BCAT2 O15382 1/20 0.37
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA9 Q16790 1/20 0.36
MEN1 O00255 2/20 0.36
KDM4E B2RXH2 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6205468 0.88 SLC6A4 (0.42) CYP2D6CCR8SLC6A2SLC6A4SLC6A3
SCHEMBL6204001 0.85 SLC6A4 (0.39) CYP2D6ATMCCR8KMT2ASLC6A2
SCHEMBL6204231 0.85 CCR8 (0.51) MAPTHPGDCCR8KMT2AHTT
SCHEMBL6411940 0.83 CCR8 (0.59) CCR8
SCHEMBL6204695 0.82 SLC6A2 (0.40) CYP2D6KMT2ASLC6A2SLC6A4SLC6A3
SCHEMBL6415241 0.82 CCR8 (0.55) MAPTCCR8KDM4E
SCHEMBL6203108 0.82 CCR8 (0.47) CCR8POLB
SCHEMBL6248463 0.81 CCR8 (0.46) MAPTHPGDCCR8KDM4E
SCHEMBL6204086 0.81 CCR8 (0.52) CCR8
SCHEMBL6256044 0.79 HTR2A (0.46) SLC6A2SLC6A4SLC6A3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1581511-A1 CCR8 INHIBITORS MILLENNIUM PHARMACEUTICALS, INC. (US) 2005-10-05 EP disclosed
WO-2004058736-A1 CCR8 INHIBITORS MILLENNIUM PHARMACEUTICALS, INC. (US) 2004-07-15 WO disclosed